Asquith CRM - Search Results

1

Discovery and Optimization of Narrow Spectrum Inhibitors of Tousled Like Kinase 2 (TLK2) Using Quantitative Structure Activity Relationships.

Asquith CRM, East MP, Laitinen T, Alamillo-Ferrer C, Hartikainen E, Wells CI, Axtman AD, Drewry DH, Tizzard GJ, Poso A, Willson TM, Johnson GL. Asquith CRM, et al. bioRxiv [Preprint]. 2023 Dec 28:2023.12.28.573261. doi: 10.1101/2023.12.28.573261. bioRxiv. 2023. Update in: Eur J Med Chem. 2024 May 5;271:116357. doi: 10.1016/j.ejmech.2024.116357. PMID: 38234837 Free PMC article. Updated. Preprint.

2

Utilizing comprehensive and mini-kinome panels to optimize the selectivity of quinoline inhibitors for cyclin G associated kinase (GAK).

Asquith CRM, Treiber DK, Zuercher WJ. Asquith CRM, et al. Bioorg Med Chem Lett. 2019 Jul 15;29(14):1727-1731. doi: 10.1016/j.bmcl.2019.05.025. Epub 2019 May 16. Bioorg Med Chem Lett. 2019. PMID: 31129055 Free article.

3

Optimization of 4-Anilinoquinolines as Dengue Virus Inhibitors.

Huang PT, Saul S, Einav S, Asquith CRM. Huang PT, et al. Among authors: asquith crm. Molecules. 2021 Dec 3;26(23):7338. doi: 10.3390/molecules26237338. Molecules. 2021. PMID: 34885921 Free PMC article.

4

Potent antiviral activity of novel multi-substituted 4-anilinoquin(az)olines.

Saul S, Pu SY, Zuercher WJ, Einav S, Asquith CRM. Saul S, et al. Among authors: asquith crm. Bioorg Med Chem Lett. 2020 Aug 15;30(16):127284. doi: 10.1016/j.bmcl.2020.127284. Epub 2020 May 27. Bioorg Med Chem Lett. 2020. PMID: 32631507

5

Identification of lead anti-human cytomegalovirus compounds targeting MAP4K4 via machine learning analysis of kinase inhibitor screening data.

Strang BL, Asquith CRM, Moshrif HF, Ho CM, Zuercher WJ, Al-Ali H. Strang BL, et al. Among authors: asquith crm. PLoS One. 2018 Jul 26;13(7):e0201321. doi: 10.1371/journal.pone.0201321. eCollection 2018. PLoS One. 2018. PMID: 30048526 Free PMC article.

6

Synthesis and Identification of Pentathiepin-Based Inhibitors of Sporothrix brasiliensis.

Asquith CRM, Machado ACS, de Miranda LHM, Konstantinova LS, Almeida-Paes R, Rakitin OA, Pereira SA. Asquith CRM, et al. Antibiotics (Basel). 2019 Dec 3;8(4):249. doi: 10.3390/antibiotics8040249. Antibiotics (Basel). 2019. PMID: 31816950 Free PMC article.

7

The Synthesis and Biological Applications of the 1,2,3-Dithiazole Scaffold.

Kalogirou AS, Oh HJ, Asquith CRM. Kalogirou AS, et al. Among authors: asquith crm. Molecules. 2023 Apr 3;28(7):3193. doi: 10.3390/molecules28073193. Molecules. 2023. PMID: 37049953 Free PMC article. Review.

8

Design and evaluation of 1,2,3-dithiazoles and fused 1,2,4-dithiazines as anti-cancer agents.

Maffuid KA, Koyioni M, Torrice CD, Murphy WA, Mewada HK, Koutentis PA, Crona DJ, Asquith CRM. Maffuid KA, et al. Among authors: asquith crm. Bioorg Med Chem Lett. 2021 Jul 1;43:128078. doi: 10.1016/j.bmcl.2021.128078. Epub 2021 May 2. Bioorg Med Chem Lett. 2021. PMID: 33951490

9

STK19: a new target for NRAS-driven cancer.

Asquith CRM, Temme L. Asquith CRM, et al. Nat Rev Drug Discov. 2020 Sep;19(9):579. doi: 10.1038/d41573-020-00116-x. Nat Rev Drug Discov. 2020. PMID: 32587355 No abstract available.

10

Novel fused tetrathiocines as antivirals that target the nucleocapsid zinc finger containing protein of the feline immunodeficiency virus (FIV) as a model of HIV infection.

Asquith CR, Meli ML, Konstantinova LS, Laitinen T, Poso A, Rakitin OA, Hofmann-Lehmann R, Allenspach K, Hilton ST. Asquith CR, et al. Bioorg Med Chem Lett. 2015 Mar 15;25(6):1352-5. doi: 10.1016/j.bmcl.2014.12.047. Epub 2014 Dec 20. Bioorg Med Chem Lett. 2015. PMID: 25702849 Free article.

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