Dehaen W - Search Results

1

Identification of novel human CC chemokine receptor 8 (CCR8) antagonists via the synthesis of naphthalene amide and sulfonamide isosteres.

Verhaegen Y, Liu L, Nguyen TT, Loy TV, Schols D, Voet ARD, Dehaen W, De Jonghe S. Verhaegen Y, et al. Among authors: dehaen w. Bioorg Chem. 2024 Apr;145:107181. doi: 10.1016/j.bioorg.2024.107181. Epub 2024 Feb 8. Bioorg Chem. 2024. PMID: 38354503

2

Synthesis and anticancer activity of novel aza-artemisinin derivatives.

Jana S, Iram S, Thomas J, Liekens S, Dehaen W. Jana S, et al. Among authors: dehaen w. Bioorg Med Chem. 2017 Jul 15;25(14):3671-3676. doi: 10.1016/j.bmc.2017.04.041. Epub 2017 Apr 30. Bioorg Med Chem. 2017. PMID: 28529044

3

Synthesis, biological evaluation and molecular modeling of a novel series of fused 1,2,3-triazoles as potential anti-coronavirus agents.

Karypidou K, Ribone SR, Quevedo MA, Persoons L, Pannecouque C, Helsen C, Claessens F, Dehaen W. Karypidou K, et al. Among authors: dehaen w. Bioorg Med Chem Lett. 2018 Nov 15;28(21):3472-3476. doi: 10.1016/j.bmcl.2018.09.019. Epub 2018 Sep 22. Bioorg Med Chem Lett. 2018. PMID: 30286952 Free PMC article.

4

Assembly of fully substituted triazolochromenes via a novel multicomponent reaction or mechanochemical synthesis.

Vroemans R, Verhaegen Y, Dieu MTT, Dehaen W. Vroemans R, et al. Among authors: dehaen w. Beilstein J Org Chem. 2018 Oct 22;14:2689-2697. doi: 10.3762/bjoc.14.246. eCollection 2018. Beilstein J Org Chem. 2018. PMID: 30410630 Free PMC article.

5

Design and synthesis of the novel oleanolic acid-cinnamic acid ester derivatives and glycyrrhetinic acid-cinnamic acid ester derivatives with cytotoxic properties.

Wang R, Yang W, Fan Y, Dehaen W, Li Y, Li H, Wang W, Zheng Q, Huai Q. Wang R, et al. Among authors: dehaen w. Bioorg Chem. 2019 Jul;88:102951. doi: 10.1016/j.bioorg.2019.102951. Epub 2019 Apr 27. Bioorg Chem. 2019. PMID: 31054427

6

Palladium-catalyzed cross-coupling reactions on a bromo-naphthalene scaffold in the search for novel human CC chemokine receptor 8 (CCR8) antagonists.

Verhaegen Y, Liu L, Nguyen TT, Van Loy T, Voet ARD, Schols D, Dehaen W, De Jonghe S. Verhaegen Y, et al. Among authors: dehaen w. Bioorg Chem. 2021 Feb;107:104560. doi: 10.1016/j.bioorg.2020.104560. Epub 2020 Dec 16. Bioorg Chem. 2021. PMID: 33383325

7

Biological characterization of ligands targeting the human CC chemokine receptor 8 (CCR8) reveals the biased signaling properties of small molecule agonists.

Liu L, Doijen J, D'huys T, Verhaegen Y, Dehaen W, De Jonghe S, Schols D, Van Loy T. Liu L, et al. Among authors: dehaen w. Biochem Pharmacol. 2021 Jun;188:114565. doi: 10.1016/j.bcp.2021.114565. Epub 2021 Apr 17. Biochem Pharmacol. 2021. PMID: 33872569 Free article.

8

Betulonic Acid Derivatives Interfering with Human Coronavirus 229E Replication via the nsp15 Endoribonuclease.

Stevaert A, Krasniqi B, Van Loy B, Nguyen T, Thomas J, Vandeput J, Jochmans D, Thiel V, Dijkman R, Dehaen W, Voet A, Naesens L. Stevaert A, et al. Among authors: dehaen w. J Med Chem. 2021 May 13;64(9):5632-5644. doi: 10.1021/acs.jmedchem.0c02124. Epub 2021 Apr 20. J Med Chem. 2021. PMID: 33877845

9

Antibacterial and antitumoral properties of 1,2,3-triazolo fused triterpenes and their mechanism of inhibiting the proliferation of HL-60 cells.

Wang R, Li Y, Hu H, Persoons L, Daelemans D, De Jonghe S, Luyten W, Krasniqi B, Dehaen W. Wang R, et al. Among authors: dehaen w. Eur J Med Chem. 2021 Nov 15;224:113727. doi: 10.1016/j.ejmech.2021.113727. Epub 2021 Jul 30. Eur J Med Chem. 2021. PMID: 34352711

10

Synthesis and Anti-HIV Activity of a Novel Series of Isoquinoline-Based CXCR4 Antagonists.

Shad MS, Claes S, Goffin E, Van Loy T, Schols D, De Jonghe S, Dehaen W. Shad MS, et al. Among authors: dehaen w. Molecules. 2021 Oct 18;26(20):6297. doi: 10.3390/molecules26206297. Molecules. 2021. PMID: 34684878 Free PMC article.

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