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Page 1
Pyrazolo[1,5-a]quinazoline scaffold as 5-deaza analogue of pyrazolo[5,1-c][1,2,4]benzotriazine system: synthesis of new derivatives, biological activity on GABAA receptor subtype and molecular dynamic study.
Guerrini G, Ciciani G, Ciattini S, Crocetti L, Daniele S, Martini C, Melani F, Vergelli C, Giovannoni MP. Guerrini G, et al. Among authors: melani f. J Enzyme Inhib Med Chem. 2016;31(2):195-204. doi: 10.3109/14756366.2015.1014475. Epub 2015 Sep 25. J Enzyme Inhib Med Chem. 2016. PMID: 25792503 Free article.
Novel 3-aroylpyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: synthesis, pharmacological and molecular modeling studies.
Guerrini G, Ciciani G, Cambi G, Bruni F, Selleri S, Melani F, Montali M, Martini C, Ghelardini C, Norcini M, Costanzo A. Guerrini G, et al. Among authors: melani f. Bioorg Med Chem. 2008 Apr 15;16(8):4471-89. doi: 10.1016/j.bmc.2008.02.058. Epub 2008 Mar 5. Bioorg Med Chem. 2008. PMID: 18325771
Synthesis, in vivo evaluation, and molecular modeling studies of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide derivatives. Identification of a bifunctional hydrogen bond area related to the inverse agonism.
Guerrini G, Ciciani G, Cambi G, Bruni F, Selleri S, Guarino C, Melani F, Montali M, Martini C, Ghelardini C, Norcini M, Costanzo A. Guerrini G, et al. Among authors: melani f. J Med Chem. 2009 Aug 13;52(15):4668-82. doi: 10.1021/jm801599a. J Med Chem. 2009. PMID: 19591485
New fluoro derivatives of the pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide system: evaluation of fluorine binding properties in the benzodiazepine site on γ-aminobutyrric acid type A (GABA(A)) receptor. Design, synthesis, biological, and molecular modeling investigation.
Guerrini G, Ciciani G, Bruni F, Selleri S, Guarino C, Melani F, Montali M, Daniele S, Martini C, Ghelardini C, Norcini M, Ciattini S, Costanzo A. Guerrini G, et al. Among authors: melani f. J Med Chem. 2010 Nov 11;53(21):7532-48. doi: 10.1021/jm1001887. J Med Chem. 2010. PMID: 20939501
New 3-, 8-disubstituted pyrazolo[5,1-c][1,2,4]benzotriazines useful for studying the interaction with the HBp-3 area (hydrogen bond point area) in the benzodiazepine site on the γ-aminobutyric acid type A (GABAA) receptor.
Guerrini G, Ciciani G, Bruni F, Selleri S, Melani F, Daniele S, Martini C, Costanzo A. Guerrini G, et al. Among authors: melani f. Bioorg Med Chem. 2011 May 15;19(10):3074-85. doi: 10.1016/j.bmc.2011.04.009. Epub 2011 Apr 12. Bioorg Med Chem. 2011. PMID: 21530274
Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: synthesis, biological evaluation and 3D-QSAR investigation.
Selleri S, Gratteri P, Costagli C, Bonaccini C, Costanzo A, Melani F, Guerrini G, Ciciani G, Costa B, Spinetti F, Martini C, Bruni F. Selleri S, et al. Among authors: melani f. Bioorg Med Chem. 2005 Aug 15;13(16):4821-34. doi: 10.1016/j.bmc.2005.05.015. Bioorg Med Chem. 2005. PMID: 15975799
178 results