Du Y - Search Results

1

Structure-Activity Relationship Studies in a Series of 2-Aryloxy-N-(pyrimidin-5-yl)acetamide Inhibitors of SLACK Potassium Channels.

Mishra NM, Spitznagel BD, Du Y, Mohamed YK, Qin Y, Weaver CD, Emmitte KA. Mishra NM, et al. Among authors: du y. Molecules. 2024 Nov 21;29(23):5494. doi: 10.3390/molecules29235494. Molecules. 2024. PMID: 39683653 Free PMC article.

2

VU0606170, a Selective Slack Channels Inhibitor, Decreases Calcium Oscillations in Cultured Cortical Neurons.

Spitznagel BD, Mishra NM, Qunies AM, Prael FJ 3rd, Du Y, Kozek KA, Lazarenko RM, Denton JS, Emmitte KA, Weaver CD. Spitznagel BD, et al. Among authors: du y. ACS Chem Neurosci. 2020 Nov 4;11(21):3658-3671. doi: 10.1021/acschemneuro.0c00583. Epub 2020 Oct 14. ACS Chem Neurosci. 2020. PMID: 33143429

3

Structure-activity relationship studies in a new series of 2-amino-N-phenylacetamide inhibitors of Slack potassium channels.

Qunies AM, Mishra NM, Spitznagel BD, Du Y, Acuña VS, David Weaver C, Emmitte KA. Qunies AM, et al. Among authors: du y. Bioorg Med Chem Lett. 2022 Nov 15;76:129013. doi: 10.1016/j.bmcl.2022.129013. Epub 2022 Sep 29. Bioorg Med Chem Lett. 2022. PMID: 36184030 Free PMC article.

4

Design, synthesis, and biological evaluation of a novel series of 1,2,4-oxadiazole inhibitors of SLACK potassium channels: Identification of in vitro tool VU0935685.

Qunies AM, Spitznagel BD, Du Y, David Weaver C, Emmitte KA. Qunies AM, et al. Among authors: du y. Bioorg Med Chem. 2023 Nov 15;95:117487. doi: 10.1016/j.bmc.2023.117487. Epub 2023 Sep 30. Bioorg Med Chem. 2023. PMID: 37812884 Free PMC article.

5

Structure-Activity Relationship Studies in a Series of Xanthine Inhibitors of SLACK Potassium Channels.

Qunies AM, Spitznagel BD, Du Y, Peprah PK, Mohamed YK, Weaver CD, Emmitte KA. Qunies AM, et al. Among authors: du y. Molecules. 2024 May 22;29(11):2437. doi: 10.3390/molecules29112437. Molecules. 2024. PMID: 38893312 Free PMC article.

6

Discovery and Characterization of VU0529331, a Synthetic Small-Molecule Activator of Homomeric G Protein-Gated, Inwardly Rectifying, Potassium (GIRK) Channels.

Kozek KA, Du Y, Sharma S, Prael FJ 3rd, Spitznagel BD, Kharade SV, Denton JS, Hopkins CR, Weaver CD. Kozek KA, et al. Among authors: du y. ACS Chem Neurosci. 2019 Jan 16;10(1):358-370. doi: 10.1021/acschemneuro.8b00287. Epub 2018 Sep 13. ACS Chem Neurosci. 2019. PMID: 30136838 Free PMC article.

7

Structure-Activity Relationship Study of the High-Affinity Neuropeptide Y₄ Receptor Positive Allosteric Modulator VU0506013.

Schüß C, Vu O, Mishra NM, Tough IR, Du Y, Stichel J, Cox HM, Weaver CD, Meiler J, Emmitte KA, Beck-Sickinger AG. Schüß C, et al. Among authors: du y. J Med Chem. 2023 Jul 13;66(13):8745-8766. doi: 10.1021/acs.jmedchem.3c00383. Epub 2023 Jun 20. J Med Chem. 2023. PMID: 37339079

8

Discovery and SAR of a novel series of GIRK1/2 and GIRK1/4 activators.

Ramos-Hunter SJ, Engers DW, Kaufmann K, Du Y, Lindsley CW, Weaver CD, Sulikowski GA. Ramos-Hunter SJ, et al. Among authors: du y. Bioorg Med Chem Lett. 2013 Sep 15;23(18):5195-8. doi: 10.1016/j.bmcl.2013.07.002. Epub 2013 Jul 18. Bioorg Med Chem Lett. 2013. PMID: 23916258 Free PMC article.

9

Development and validation of a thallium flux-based functional assay for the sodium channel NaV1.7 and its utility for lead discovery and compound profiling.

Du Y, Days E, Romaine I, Abney KK, Kaufmann K, Sulikowski G, Stauffer S, Lindsley CW, Weaver CD. Du Y, et al. ACS Chem Neurosci. 2015 Jun 17;6(6):871-8. doi: 10.1021/acschemneuro.5b00004. Epub 2015 Apr 30. ACS Chem Neurosci. 2015. PMID: 25879403

10

Highly Selective Y₄ Receptor Antagonist Binds in an Allosteric Binding Pocket.

Schüß C, Vu O, Schubert M, Du Y, Mishra NM, Tough IR, Stichel J, Weaver CD, Emmitte KA, Cox HM, Meiler J, Beck-Sickinger AG. Schüß C, et al. Among authors: du y. J Med Chem. 2021 Mar 11;64(5):2801-2814. doi: 10.1021/acs.jmedchem.0c02000. Epub 2021 Feb 17. J Med Chem. 2021. PMID: 33595306

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