Carrupt PA - Search Results

1

Inhibition of monoamine oxidase-B by 5H-indeno[1,2-c]pyridazines: biological activities, quantitative structure-activity relationships (QSARs) and 3D-QSARs.

Kneubühler S, Thull U, Altomare C, Carta V, Gaillard P, Carrupt PA, Carotti A, Testa B. Kneubühler S, et al. Among authors: carrupt pa. J Med Chem. 1995 Sep 15;38(19):3874-83. doi: 10.1021/jm00019a018. J Med Chem. 1995. PMID: 7562919

2

Human recombinant monoamine oxidase B as reliable and efficient enzyme source for inhibitor screening.

Novaroli L, Reist M, Favre E, Carotti A, Catto M, Carrupt PA. Novaroli L, et al. Among authors: carrupt pa. Bioorg Med Chem. 2005 Nov 15;13(22):6212-7. doi: 10.1016/j.bmc.2005.06.043. Epub 2005 Jul 27. Bioorg Med Chem. 2005. PMID: 16054369

3

Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases.

Farina R, Pisani L, Catto M, Nicolotti O, Gadaleta D, Denora N, Soto-Otero R, Mendez-Alvarez E, Passos CS, Muncipinto G, Altomare CD, Nurisso A, Carrupt PA, Carotti A. Farina R, et al. Among authors: carrupt pa. J Med Chem. 2015 Jul 23;58(14):5561-78. doi: 10.1021/acs.jmedchem.5b00599. Epub 2015 Jul 9. J Med Chem. 2015. PMID: 26107513

4

Quantitative structure-metabolism relationship analyses of MAO-mediated toxication of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine and analogues.

Altomare C, Carrupt PA, Gaillard P, el Tayar N, Testa B, Carotti A. Altomare C, et al. Among authors: carrupt pa. Chem Res Toxicol. 1992 May-Jun;5(3):366-75. doi: 10.1021/tx00027a008. Chem Res Toxicol. 1992. PMID: 1504260

5

Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists.

el Tayar N, Carrupt PA, Van de Waterbeemd H, Testa B. el Tayar N, et al. Among authors: carrupt pa. J Med Chem. 1988 Nov;31(11):2072-81. doi: 10.1021/jm00119a004. J Med Chem. 1988. PMID: 2903243 Review.

6

Inhibition of monoamine oxidase by isoquinoline derivatives. Qualitative and 3D-quantitative structure-activity relationships.

Thull U, Kneubühler S, Gaillard P, Carrupt PA, Testa B, Altomare C, Carotti A, Jenner P, McNaught KS. Thull U, et al. Among authors: carrupt pa. Biochem Pharmacol. 1995 Sep 7;50(6):869-77. doi: 10.1016/0006-2952(95)00220-t. Biochem Pharmacol. 1995. PMID: 7575650

7

Molecular lipophilicity potential, a tool in 3D QSAR: method and applications.

Gaillard P, Carrupt PA, Testa B, Boudon A. Gaillard P, et al. Among authors: carrupt pa. J Comput Aided Mol Des. 1994 Apr;8(2):83-96. doi: 10.1007/BF00119860. J Comput Aided Mol Des. 1994. PMID: 7914913

8

Effects of solvation on the ionization and conformation of raclopride and other antidopaminergic 6-methoxysalicylamides: insight into the pharmacophore.

Tsai RS, Carrupt PA, Testa B, Gaillard P, el Tayar N, Högberg T. Tsai RS, et al. Among authors: carrupt pa. J Med Chem. 1993 Jan 22;36(2):196-204. doi: 10.1021/jm00054a002. J Med Chem. 1993. PMID: 8423592

9

Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.

Gaillard P, Carrupt PA, Testa B, Schambel P. Gaillard P, et al. Among authors: carrupt pa. J Med Chem. 1996 Jan 5;39(1):126-34. doi: 10.1021/jm950410b. J Med Chem. 1996. PMID: 8568799

10

Inhibition of monoamine oxidase-B by condensed pyridazines and pyrimidines: effects of lipophilicity and structure-activity relationships.

Altomare C, Cellamare S, Summo L, Catto M, Carotti A, Thull U, Carrupt PA, Testa B, Stoeckli-Evans H. Altomare C, et al. Among authors: carrupt pa. J Med Chem. 1998 Sep 24;41(20):3812-20. doi: 10.1021/jm981005y. J Med Chem. 1998. PMID: 9748356

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