Goldman ME - Search Results

1

5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.

Williams TM, Ciccarone TM, MacTough SC, Rooney CS, Balani SK, Condra JH, Emini EA, Goldman ME, Greenlee WJ, Kauffman LR, et al. Williams TM, et al. Among authors: goldman me. J Med Chem. 1993 Apr 30;36(9):1291-4. doi: 10.1021/jm00061a022. J Med Chem. 1993. PMID: 7683725

2

Synthesis and evaluation of 2-pyridinone derivatives as HIV-1-specific reverse transcriptase inhibitors. 2. Analogues of 3-aminopyridin-2(1H)-one.

Saari WS, Wai JS, Fisher TE, Thomas CM, Hoffman JM, Rooney CS, Smith AM, Jones JH, Bamberger DL, Goldman ME, et al. Saari WS, et al. Among authors: goldman me. J Med Chem. 1992 Oct 16;35(21):3792-802. doi: 10.1021/jm00099a007. J Med Chem. 1992. PMID: 1279173

3

Metabolism of a new HIV-1 reverse transcriptase inhibitor, 3-[2-(benzoxazol-2-yl)ethyl]-5-ethyl-6-methylpyridin-2(1H)-one (L-696,229), in rat and liver slices.

Balani SK, Pitzenberger SM, Kauffman LR, Arison BH, Ramjit HG, Goldman ME, O'Brien JA, King JD, Hoffman JM, Rooney CS, et al. Balani SK, et al. Among authors: goldman me. Drug Metab Dispos. 1992 Nov-Dec;20(6):869-76. Drug Metab Dispos. 1992. PMID: 1283569

4

2-Pyridinone derivatives: a new class of nonnucleoside, HIV-1-specific reverse transcriptase inhibitors.

Saari WS, Hoffman JM, Wai JS, Fisher TE, Rooney CS, Smith AM, Thomas CM, Goldman ME, O'Brien JA, Nunberg JH, et al. Saari WS, et al. Among authors: goldman me. J Med Chem. 1991 Sep;34(9):2922-5. doi: 10.1021/jm00113a036. J Med Chem. 1991. PMID: 1716683 No abstract available.

5

Metabolism of 3-[2-(benzoxazol-2-yl)ethyl]-5-ethyl-6-methylpyridin-2 (1H)-one (L-696,229), an HIV-1 reverse transcriptase inhibitor, by rat liver slices and in humans.

Balani SK, Kauffman LR, Arison BH, Olah TV, Goldman ME, Varga SL, O'Brien JA, Ramjit HG, Rooney CS, Hoffman JM, et al. Balani SK, et al. Among authors: goldman me. Drug Metab Dispos. 1994 Mar-Apr;22(2):200-5. Drug Metab Dispos. 1994. PMID: 7516852

6

A nonnucleoside reverse transcriptase inhibitor active on human immunodeficiency virus type 1 isolates resistant to related inhibitors.

Goldman ME, O'Brien JA, Ruffing TL, Schleif WA, Sardana VV, Byrnes VW, Condra JH, Hoffman JM, Emini EA. Goldman ME, et al. Antimicrob Agents Chemother. 1993 May;37(5):947-9. doi: 10.1128/AAC.37.5.947. Antimicrob Agents Chemother. 1993. PMID: 7685996 Free PMC article.

7

Biotransformation of 5-chloro-3-phenylthioindole-2-carboxamide (L-734,005) in rhesus monkeys and rat liver microsomes to a potent HIV-1 reverse transcriptase inhibitor.

Balani SK, Goldman ME, Kauffman LR, Varga SL, O'Brien JA, Smith SJ, Olah TV, Ramjit HG, Schorn TW, Pitzenberger SM, et al. Balani SK, et al. Among authors: goldman me. Drug Metab Dispos. 1993 Jul-Aug;21(4):598-604. Drug Metab Dispos. 1993. PMID: 7690697

8

L-696,229 specifically inhibits human immunodeficiency virus type 1 reverse transcriptase and possesses antiviral activity in vitro.

Goldman ME, O'Brien JA, Ruffing TL, Nunberg JH, Schleif WA, Quintero JC, Siegl PK, Hoffman JM, Smith AM, Emini EA. Goldman ME, et al. Antimicrob Agents Chemother. 1992 May;36(5):1019-23. doi: 10.1128/AAC.36.5.1019. Antimicrob Agents Chemother. 1992. PMID: 1380788 Free PMC article.

9

Inhibition of human immunodeficiency virus-1 reverse transcriptase activity by rubromycins: competitive interaction at the template.primer site.

Goldman ME, Salituro GS, Bowen JA, Williamson JM, Zink DL, Schleif WA, Emini EA. Goldman ME, et al. Mol Pharmacol. 1990 Jul;38(1):20-5. Mol Pharmacol. 1990. PMID: 1695317

10

Viral resistance to human immunodeficiency virus type 1-specific pyridinone reverse transcriptase inhibitors.

Nunberg JH, Schleif WA, Boots EJ, O'Brien JA, Quintero JC, Hoffman JM, Emini EA, Goldman ME. Nunberg JH, et al. Among authors: goldman me. J Virol. 1991 Sep;65(9):4887-92. doi: 10.1128/JVI.65.9.4887-4892.1991. J Virol. 1991. PMID: 1714522 Free PMC article.

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