Ellsworth K - Search Results

1

4,7 beta-Dimethyl-4-azacholestan-3-one (MK-386) and related 4-azasteroids as selective inhibitors of human type 1 5 alpha-reductase.

Bakshi RK, Patel GF, Rasmusson GH, Baginsky WF, Cimis G, Ellsworth K, Chang B, Bull H, Tolman RL, Harris GS. Bakshi RK, et al. Among authors: ellsworth k. J Med Chem. 1994 Nov 11;37(23):3871-4. doi: 10.1021/jm00049a003. J Med Chem. 1994. PMID: 7966146 No abstract available.

2

Identification and selective inhibition of an isozyme of steroid 5 alpha-reductase in human scalp.

Harris G, Azzolina B, Baginsky W, Cimis G, Rasmusson GH, Tolman RL, Raetz CR, Ellsworth K. Harris G, et al. Among authors: ellsworth k. Proc Natl Acad Sci U S A. 1992 Nov 15;89(22):10787-91. doi: 10.1073/pnas.89.22.10787. Proc Natl Acad Sci U S A. 1992. PMID: 1438277 Free PMC article.

3

4-Aza-3-oxo-5 alpha-androst-1-ene-17 beta-N-aryl-carboxamides as dual inhibitors of human type 1 and type 2 steroid 5 alpha-reductases. Dramatic effect of N-aryl substituents on type 1 and type 2 5 alpha-reductase inhibitory potency.

Bakshi RK, Rasmusson GH, Patel GF, Mosley RT, Chang B, Ellsworth K, Harris GS, Tolman RL. Bakshi RK, et al. Among authors: ellsworth k. J Med Chem. 1995 Aug 18;38(17):3189-92. doi: 10.1021/jm00017a001. J Med Chem. 1995. PMID: 7650670 No abstract available.

4

MK386: a potent, selective inhibitor of the human type 1 5alpha-reductase.

Ellsworth K, Azzolina B, Baginsky W, Bull H, Chang B, Cimis G, Mitra S, Toney J, Bakshi RK, Rasmusson GR, Tolman RL, Harris GS. Ellsworth K, et al. J Steroid Biochem Mol Biol. 1996 Jul;58(4):377-84. doi: 10.1016/0960-0760(96)00050-7. J Steroid Biochem Mol Biol. 1996. PMID: 8903421

5

Novel 3,4-dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase a.

Rosauer KG, Ogawa AK, Willoughby CA, Ellsworth KP, Geissler WM, Myers RW, Deng Q, Chapman KT, Harris G, Moller DE. Rosauer KG, et al. Among authors: ellsworth kp. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4385-8. doi: 10.1016/j.bmcl.2003.09.022. Bioorg Med Chem Lett. 2003. PMID: 14643331

6

Cloning, expression and characterization of rhesus macaque types 1 and 2 5alpha-reductase: evidence for mechanism-based inhibition by finasteride.

Ellsworth KP, Azzolina BA, Cimis G, Bull HG, Harris GS. Ellsworth KP, et al. J Steroid Biochem Mol Biol. 1998 Sep;66(5-6):271-9. doi: 10.1016/s0960-0760(98)00059-4. J Steroid Biochem Mol Biol. 1998. PMID: 9749833

7

Expression of the type 1 and 2 steroid 5 alpha-reductases in human fetal tissues.

Ellsworth K, Harris G. Ellsworth K, et al. Biochem Biophys Res Commun. 1995 Oct 13;215(2):774-80. doi: 10.1006/bbrc.1995.2530. Biochem Biophys Res Commun. 1995. PMID: 7488021

8

Inhibition of rat alpha-reductases by finasteride: evidence for isozyme differences in the mechanism of inhibition.

Azzolina B, Ellsworth K, Andersson S, Geissler W, Bull HG, Harris GS. Azzolina B, et al. Among authors: ellsworth k. J Steroid Biochem Mol Biol. 1997 Apr;61(1-2):55-64. doi: 10.1016/s0960-0760(97)00002-2. J Steroid Biochem Mol Biol. 1997. PMID: 9328210

9

Design and synthesis of novel antibacterial agents with inhibitory activity against DNA polymerase III.

Ali A, Aster SD, Graham DW, Patel GF, Taylor GE, Tolman RL, Painter RE, Silver LL, Young K, Ellsworth K, Geissler W, Harris GS. Ali A, et al. Among authors: ellsworth k. Bioorg Med Chem Lett. 2001 Aug 20;11(16):2185-8. doi: 10.1016/s0960-894x(01)00407-3. Bioorg Med Chem Lett. 2001. PMID: 11514166

10

Novel pyrazolo[3,4-d]pyrimidine-based inhibitors of Staphlococcus aureus DNA polymerase III: design, synthesis, and biological evaluation.

Ali A, Taylor GE, Ellsworth K, Harris G, Painter R, Silver LL, Young K. Ali A, et al. Among authors: ellsworth k. J Med Chem. 2003 May 8;46(10):1824-30. doi: 10.1021/jm020483c. J Med Chem. 2003. PMID: 12723946

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

83 results

Search Page

Filters