Mederski WW - Search Results

1

Non-peptide angiotensin II receptor antagonists: synthesis and biological activity of a series of novel 4,5-dihydro-4-oxo-3H-imidazo[4,5-c]pyridine derivatives.

Mederski WW, Dorsch D, Bokel HH, Beier N, Lues I, Schelling P. Mederski WW, et al. J Med Chem. 1994 May 27;37(11):1632-45. doi: 10.1021/jm00037a014. J Med Chem. 1994. PMID: 8201597

2

Endothelin antagonists: discovery of EMD 122946, a highly potent and orally active ETA selective antagonist.

Mederski WW, Dorsch D, Osswald M, Anzali S, Christadler M, Schmitges CJ, Schelling P, Wilm C, Fluck M. Mederski WW, et al. Bioorg Med Chem Lett. 1998 Jul 7;8(13):1771-6. doi: 10.1016/s0960-894x(98)00301-1. Bioorg Med Chem Lett. 1998. PMID: 9873432

3

Benzofuro[3,2-b]pyridines as mixed ET(A)/ET(B) and selective ET(B) endothelin receptor antagonists.

Mederski WW, Osswald M, Dorsch D, Christadler M, Schmitges CJ, Wilm C. Mederski WW, et al. Bioorg Med Chem Lett. 1999 Feb 22;9(4):619-22. doi: 10.1016/s0960-894x(99)00040-2. Bioorg Med Chem Lett. 1999. PMID: 10098676

4

Halothiophene benzimidazoles as P1 surrogates of inhibitors of blood coagulation factor Xa.

Mederski WW, Dorsch D, Anzali S, Gleitz J, Cezanne B, Tsaklakidis C. Mederski WW, et al. Bioorg Med Chem Lett. 2004 Jul 16;14(14):3763-9. doi: 10.1016/j.bmcl.2004.04.097. Bioorg Med Chem Lett. 2004. PMID: 15203158

5

Chlorothiophenecarboxamides as P1 surrogates of inhibitors of blood coagulation factor Xa.

Mederski WW, Cezanne B, van Amsterdam C, Bühring KU, Dorsch D, Gleitz J, März J, Tsaklakidis C. Mederski WW, et al. Bioorg Med Chem Lett. 2004 Dec 6;14(23):5817-22. doi: 10.1016/j.bmcl.2004.09.043. Bioorg Med Chem Lett. 2004. PMID: 15501047

6

Endothelin antagonists: search for surrogates of methylendioxyphenyl by means of a Kohonen neural network.

Anzali S, Mederski WW, Osswald M, Dorsch D. Anzali S, et al. Among authors: mederski ww. Bioorg Med Chem Lett. 1998 Jan 6;8(1):11-6. doi: 10.1016/s0960-894x(97)10150-0. Bioorg Med Chem Lett. 1998. PMID: 9871620

7

Endothelin antagonists: evaluation of 2,1,3-benzothiadiazole as a methylendioxyphenyl bioisoster.

Mederski WW, Osswald M, Dorsch D, Anzali S, Christadler M, Schmitges CJ, Wilm C. Mederski WW, et al. Bioorg Med Chem Lett. 1998 Jan 6;8(1):17-22. doi: 10.1016/s0960-894x(97)10151-2. Bioorg Med Chem Lett. 1998. PMID: 9871621

8

pH-dependent binding modes observed in trypsin crystals: lessons for structure-based drug design.

Stubbs MT, Reyda S, Dullweber F, Möller M, Klebe G, Dorsch D, Mederski WW, Wurziger H. Stubbs MT, et al. Among authors: mederski ww. Chembiochem. 2002 Mar 1;3(2-3):246-9. doi: 10.1002/1439-7633(20020301)3:2/3<246::aid-cbic246>3.0.co;2-#. Chembiochem. 2002. PMID: 11921406 No abstract available.

9

A general synthesis of 1-aryl carbamoyl-2-alkyl-4-aryl substituted semicarbazides as nonbasic factor Xa inhibitors.

Mederski WW, Germann M. Mederski WW, et al. Bioorg Med Chem Lett. 2003 Nov 3;13(21):3715-8. doi: 10.1016/j.bmcl.2003.08.007. Bioorg Med Chem Lett. 2003. PMID: 14552764

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