Felock PJ - Search Results

1

The role of manganese in promoting multimerization and assembly of human immunodeficiency virus type 1 integrase as a catalytically active complex on immobilized long terminal repeat substrates.

Wolfe AL, Felock PJ, Hastings JC, Blau CU, Hazuda DJ. Wolfe AL, et al. Among authors: felock pj. J Virol. 1996 Mar;70(3):1424-32. doi: 10.1128/JVI.70.3.1424-1432.1996. J Virol. 1996. PMID: 8627659 Free PMC article.

2

Equivalent inhibition of half-site and full-site retroviral strand transfer reactions by structurally diverse compounds.

Hazuda D, Felock P, Hastings J, Pramanik B, Wolfe A, Goodarzi G, Vora A, Brackmann K, Grandgenett D. Hazuda D, et al. J Virol. 1997 Jan;71(1):807-11. doi: 10.1128/JVI.71.1.807-811.1997. J Virol. 1997. PMID: 8985421 Free PMC article.

3

Isolation and characterization of novel human immunodeficiency virus integrase inhibitors from fungal metabolites.

Hazuda D, Blau CU, Felock P, Hastings J, Pramanik B, Wolfe A, Bushman F, Farnet C, Goetz M, Williams M, Silverman K, Lingham R, Singh S. Hazuda D, et al. Antivir Chem Chemother. 1999 Mar;10(2):63-70. doi: 10.1177/095632029901000202. Antivir Chem Chemother. 1999. PMID: 10335400 Free article.

4

Inhibitors of strand transfer that prevent integration and inhibit HIV-1 replication in cells.

Hazuda DJ, Felock P, Witmer M, Wolfe A, Stillmock K, Grobler JA, Espeseth A, Gabryelski L, Schleif W, Blau C, Miller MD. Hazuda DJ, et al. Science. 2000 Jan 28;287(5453):646-50. doi: 10.1126/science.287.5453.646. Science. 2000. PMID: 10649997

5

HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase.

Espeseth AS, Felock P, Wolfe A, Witmer M, Grobler J, Anthony N, Egbertson M, Melamed JY, Young S, Hamill T, Cole JL, Hazuda DJ. Espeseth AS, et al. Proc Natl Acad Sci U S A. 2000 Oct 10;97(21):11244-9. doi: 10.1073/pnas.200139397. Proc Natl Acad Sci U S A. 2000. PMID: 11016953 Free PMC article.

6

Differential divalent cation requirements uncouple the assembly and catalytic reactions of human immunodeficiency virus type 1 integrase.

Hazuda DJ, Felock PJ, Hastings JC, Pramanik B, Wolfe AL. Hazuda DJ, et al. Among authors: felock pj. J Virol. 1997 Sep;71(9):7005-11. doi: 10.1128/JVI.71.9.7005-7011.1997. J Virol. 1997. PMID: 9261430 Free PMC article.

7

Discovery and analysis of inhibitors of the human immunodeficiency integrase.

Hazuda D, Felock PJ, Hastings JC, Pramanik B, Wolfe AL. Hazuda D, et al. Among authors: felock pj. Drug Des Discov. 1997 May;15(1):17-24. Drug Des Discov. 1997. PMID: 9332828

8

Design and synthesis of 8-hydroxy-[1,6]naphthyridines as novel inhibitors of HIV-1 integrase in vitro and in infected cells.

Zhuang L, Wai JS, Embrey MW, Fisher TE, Egbertson MS, Payne LS, Guare JP Jr, Vacca JP, Hazuda DJ, Felock PJ, Wolfe AL, Stillmock KA, Witmer MV, Moyer G, Schleif WA, Gabryelski LJ, Leonard YM, Lynch JJ Jr, Michelson SR, Young SD. Zhuang L, et al. Among authors: felock pj. J Med Chem. 2003 Feb 13;46(4):453-6. doi: 10.1021/jm025553u. J Med Chem. 2003. PMID: 12570367

9

A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase.

Hazuda DJ, Anthony NJ, Gomez RP, Jolly SM, Wai JS, Zhuang L, Fisher TE, Embrey M, Guare JP Jr, Egbertson MS, Vacca JP, Huff JR, Felock PJ, Witmer MV, Stillmock KA, Danovich R, Grobler J, Miller MD, Espeseth AS, Jin L, Chen IW, Lin JH, Kassahun K, Ellis JD, Wong BK, Xu W, Pearson PG, Schleif WA, Cortese R, Emini E, Summa V, Holloway MK, Young SD. Hazuda DJ, et al. Among authors: felock pj. Proc Natl Acad Sci U S A. 2004 Aug 3;101(31):11233-8. doi: 10.1073/pnas.0402357101. Epub 2004 Jul 26. Proc Natl Acad Sci U S A. 2004. PMID: 15277684 Free PMC article.

10

Design and synthesis of substituted 4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamides, novel HIV-1 integrase inhibitors.

Langford HM, Williams PD, Homnick CF, Vacca JP, Felock PJ, Stillmock KA, Witmer MV, Hazuda DJ, Gabryelski LJ, Schleif WA. Langford HM, et al. Among authors: felock pj. Bioorg Med Chem Lett. 2008 Jan 15;18(2):721-5. doi: 10.1016/j.bmcl.2007.11.049. Epub 2007 Nov 19. Bioorg Med Chem Lett. 2008. PMID: 18078751

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