Bryant SD - Search Results

1

Opioid receptor selectivity alteration by single residue replacement: synthesis and activity profile of [Dmt1]deltorphin B.

Guerrini R, Capasso A, Sorrentino L, Anacardio R, Bryant SD, Lazarus LH, Attila M, Salvadori S. Guerrini R, et al. Among authors: bryant sd. Eur J Pharmacol. 1996 Apr 29;302(1-3):37-42. doi: 10.1016/0014-2999(96)00067-2. Eur J Pharmacol. 1996. PMID: 8790989

2

Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors.

Salvadori S, Bryant SD, Bianchi C, Balboni G, Scaranari V, Attila M, Lazarus LH. Salvadori S, et al. Among authors: bryant sd. J Med Chem. 1993 Nov 26;36(24):3748-56. doi: 10.1021/jm00076a001. J Med Chem. 1993. PMID: 8254604

3

Relationship between receptor affinity and topography of N-terminally extended and bridged [Tyr1-->Asp4]deltorphin C analogues: novel probes for the delta-opioid receptor.

Salvadori S, Bryant SD, Temussi PA, Bundy DM, Attila M, Tomatis R, Lazarus LH. Salvadori S, et al. Among authors: bryant sd. Eur J Pharmacol. 1993 Jan 19;230(3):357-61. doi: 10.1016/0014-2999(93)90573-z. Eur J Pharmacol. 1993. PMID: 8382619

4

Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.

Salvadori S, Attila M, Balboni G, Bianchi C, Bryant SD, Crescenzi O, Guerrini R, Picone D, Tancredi T, Temussi PA, et al. Salvadori S, et al. Among authors: bryant sd. Mol Med. 1995 Sep;1(6):678-89. Mol Med. 1995. PMID: 8529134 Free PMC article.

5

Design and synthesis of 1-aminocycloalkane-1-carboxylic acid-substituted deltorphin analogues: unique delta and mu opioid activity in modified peptides.

Breveglieri A, Guerrini R, Salvadori S, Bianchi C, Bryant SD, Attila M, Lazarus LH. Breveglieri A, et al. Among authors: bryant sd. J Med Chem. 1996 Feb 2;39(3):773-80. doi: 10.1021/jm950490j. J Med Chem. 1996. PMID: 8576920

6

Dmt-Tic-OH a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse.

Capasso A, Guerrini R, Balboni G, Sorrentino L, Temussi P, Lazarus LH, Bryant SD, Salvadori S. Capasso A, et al. Among authors: bryant sd. Life Sci. 1996;59(8):PL93-8. doi: 10.1016/0024-3205(96)00353-0. Life Sci. 1996. PMID: 8761022

7

Opioid diketopiperazines: synthesis and activity of a prototypic class of opioid antagonists.

Balboni G, Guerrini R, Salvadori S, Tomatis R, Bryant SD, Bianchi C, Attila M, Lazarus LH. Balboni G, et al. Among authors: bryant sd. Biol Chem. 1997 Jan;378(1):19-29. doi: 10.1515/bchm.1997.378.1.19. Biol Chem. 1997. PMID: 9049061

8

Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary delta opioid antagonist activity.

Salvadori S, Balboni G, Guerrini R, Tomatis R, Bianchi C, Bryant SD, Cooper PS, Lazarus LH. Salvadori S, et al. Among authors: bryant sd. J Med Chem. 1997 Sep 12;40(19):3100-8. doi: 10.1021/jm9607663. J Med Chem. 1997. PMID: 9301674

9

Rational design of dynorphin A analogues with delta-receptor selectivity and antagonism for delta- and kappa-receptors.

Guerrini R, Capasso A, Marastoni M, Bryant SD, Cooper PS, Lazarus LH, Temussi PA, Salvadori S. Guerrini R, et al. Among authors: bryant sd. Bioorg Med Chem. 1998 Jan;6(1):57-62. doi: 10.1016/s0968-0896(97)10008-6. Bioorg Med Chem. 1998. PMID: 9502105

10

Further studies on the Dmt-Tic pharmacophore: hydrophobic substituents at the C-terminus endow delta antagonists to manifest mu agonism or mu antagonism.

Salvadori S, Guerrini R, Balboni G, Bianchi C, Bryant SD, Cooper PS, Lazarus LH. Salvadori S, et al. Among authors: bryant sd. J Med Chem. 1999 Dec 2;42(24):5010-9. doi: 10.1021/jm990165m. J Med Chem. 1999. PMID: 10585210

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