Scozzafava A - Search Results

1

Carbonic anhydrase activators: X-ray crystallographic and spectroscopic investigations for the interaction of isozymes I and II with histamine.

Briganti F, Mangani S, Orioli P, Scozzafava A, Vernaglione G, Supuran CT. Briganti F, et al. Among authors: scozzafava a. Biochemistry. 1997 Aug 26;36(34):10384-92. doi: 10.1021/bi970760v. Biochemistry. 1997. PMID: 9265618

2

Carbonic anhydrase activators: high affinity isozymes I, II, and IV activators, incorporating a beta-alanyl-histidine scaffold.

Scozzafava A, Supuran CT. Scozzafava A, et al. J Med Chem. 2002 Jan 17;45(2):284-91. doi: 10.1021/jm010958k. J Med Chem. 2002. PMID: 11784133

3

Carbonic anhydrase activators: human isozyme II is strongly activated by oligopeptides incorporating the carboxyterminal sequence of the bicarbonate anion exchanger AE1.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem Lett. 2002 Apr 22;12(8):1177-80. doi: 10.1016/s0960-894x(02)00121-x. Bioorg Med Chem Lett. 2002. PMID: 11934582

4

Crystal structure of a zinc-activated variant of human carbonic anhydrase I, CA I Michigan 1: evidence for a second zinc binding site involving arginine coordination.

Ferraroni M, Tilli S, Briganti F, Chegwidden WR, Supuran CT, Wiebauer KE, Tashian RE, Scozzafava A. Ferraroni M, et al. Among authors: scozzafava a. Biochemistry. 2002 May 21;41(20):6237-44. doi: 10.1021/bi0120446. Biochemistry. 2002. PMID: 12009884

5

Nonaromatic sulfonamide group as an ideal anchor for potent human carbonic anhydrase inhibitors: role of hydrogen-bonding networks in ligand binding and drug design.

Abbate F, Supuran CT, Scozzafava A, Orioli P, Stubbs MT, Klebe G. Abbate F, et al. Among authors: scozzafava a. J Med Chem. 2002 Aug 15;45(17):3583-7. doi: 10.1021/jm011131t. J Med Chem. 2002. PMID: 12166931

6

Hydroxyurea is a carbonic anhydrase inhibitor.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem. 2003 May 15;11(10):2241-6. doi: 10.1016/s0968-0896(03)00112-3. Bioorg Med Chem. 2003. PMID: 12713833

7

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one?

Casini A, Abbate F, Scozzafava A, Supuran CT. Casini A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2003 Aug 18;13(16):2759-63. doi: 10.1016/s0960-894x(03)00508-0. Bioorg Med Chem Lett. 2003. PMID: 12873509

8

Carbonic anhydrase activators. The selective serotonin reuptake inhibitors fluoxetine, sertraline and citalopram are strong activators of isozymes I and II.

Casini A, Caccia S, Scozzafava A, Supuran CT. Casini A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2003 Aug 18;13(16):2765-8. doi: 10.1016/s0960-894x(03)00507-9. Bioorg Med Chem Lett. 2003. PMID: 12873510

9

Design of weakly basic thrombin inhibitors incorporating novel P1 binding functions: molecular and X-ray crystallographic studies.

De Simone G, Menchise V, Omaggio S, Pedone C, Scozzafava A, Supuran CT. De Simone G, et al. Among authors: scozzafava a. Biochemistry. 2003 Aug 5;42(30):9013-21. doi: 10.1021/bi020512l. Biochemistry. 2003. PMID: 12885234

10

Designing of novel carbonic anhydrase inhibitors and activators.

Supuran CT, Vullo D, Manole G, Casini A, Scozzafava A. Supuran CT, et al. Among authors: scozzafava a. Curr Med Chem Cardiovasc Hematol Agents. 2004 Jan;2(1):49-68. Curr Med Chem Cardiovasc Hematol Agents. 2004. PMID: 15328829 Review.

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