Krushinski J - Search Results

1

N-Methyl-5-tert-butyltryptamine: A novel, highly potent 5-HT1D receptor agonist.

Xu YC, Schaus JM, Walker C, Krushinski J, Adham N, Zgombick JM, Liang SX, Kohlman DT, Audia JE. Xu YC, et al. Among authors: krushinski j. J Med Chem. 1999 Feb 11;42(3):526-31. doi: 10.1021/jm9805945. J Med Chem. 1999. PMID: 9986723

2

Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists.

Zhang D, Kohlman D, Krushinski J, Liang S, Ying BP, Reilly JE, Dinn SR, Wainscott DB, Nutter S, Gough W, Nelson DL, Schaus JM, Xu YC. Zhang D, et al. Among authors: krushinski j. Bioorg Med Chem Lett. 2004 Dec 20;14(24):6011-6. doi: 10.1016/j.bmcl.2004.09.079. Bioorg Med Chem Lett. 2004. PMID: 15546719

3

Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT₁ F receptor agonists: Evolution from bicyclic to monocyclic cores.

Zhang D, Blanco MJ, Ying BP, Kohlman D, Liang SX, Victor F, Chen Q, Krushinski J, Filla SA, Hudziak KJ, Mathes BM, Cohen MP, Zacherl D, Nelson DL, Wainscott DB, Nutter SE, Gough WH, Schaus JM, Xu YC. Zhang D, et al. Among authors: krushinski j. Bioorg Med Chem Lett. 2015 Oct 1;25(19):4337-41. doi: 10.1016/j.bmcl.2015.07.042. Epub 2015 Jul 22. Bioorg Med Chem Lett. 2015. PMID: 26271587

4

[3H]LY334370, a novel radioligand for the 5-HT1F receptor. I. In vitro characterization of binding properties.

Wainscott DB, Krushinski JH Jr, Audia JE, Schaus JM, Zgombick JM, Lucaites VL, Nelson DL. Wainscott DB, et al. Naunyn Schmiedebergs Arch Pharmacol. 2005 Mar;371(3):169-77. doi: 10.1007/s00210-005-1035-9. Epub 2005 Apr 27. Naunyn Schmiedebergs Arch Pharmacol. 2005. PMID: 15900510

5

[3H]LY334370, a novel radioligand for the 5-HT1F receptor. II. Autoradiographic localization in rat, guinea pig, monkey and human brain.

Lucaites VL, Krushinski JH, Schaus JM, Audia JE, Nelson DL. Lucaites VL, et al. Naunyn Schmiedebergs Arch Pharmacol. 2005 Mar;371(3):178-84. doi: 10.1007/s00210-005-1036-8. Epub 2005 Apr 27. Naunyn Schmiedebergs Arch Pharmacol. 2005. PMID: 15900511

6

Indoloxypropanolamine analogues as 5-HT(1A) receptor antagonists.

Krushinski JH Jr, Schaus JM, Thompson DC, Calligaro DO, Nelson DL, Luecke SH, Wainscott DB, Wong DT. Krushinski JH Jr, et al. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5600-4. doi: 10.1016/j.bmcl.2007.07.086. Epub 2007 Aug 22. Bioorg Med Chem Lett. 2007. PMID: 17804228

7

Synthesis, ex vivo evaluation, and radiolabeling of potent 1,5-diphenylpyrrolidin-2-one cannabinoid subtype-1 receptor ligands as candidates for in vivo imaging.

Donohue SR, Krushinski JH, Pike VW, Chernet E, Phebus L, Chesterfield AK, Felder CC, Halldin C, Schaus JM. Donohue SR, et al. Among authors: krushinski jh. J Med Chem. 2008 Sep 25;51(18):5833-42. doi: 10.1021/jm800416m. J Med Chem. 2008. PMID: 18800770 Free PMC article.

8

3-Aryl-1,2-diacetamidopropane derivatives as novel and potent NK-1 receptor antagonists.

Hipskind PA, Howbert JJ, Bruns RF, Cho SS, Crowell TA, Foreman MM, Gehlert DR, Iyengar S, Johnson KW, Krushinski JH, Li DL, Lobb KL, Mason NR, Muehl BS, Nixon JA, Phebus LA, Regoli D, Simmons RM, Threlkeld PG, Waters DC, Gitter BD. Hipskind PA, et al. Among authors: krushinski jh. J Med Chem. 1996 Feb 2;39(3):736-48. doi: 10.1021/jm950616c. J Med Chem. 1996. PMID: 8576917

9

Pharmacological characterization of the cannabinoid CB₁ receptor PET ligand ortholog, [³H]MePPEP.

Suter TM, Chesterfield AK, Bao C, Schaus JM, Krushinski JH, Statnick MA, Felder CC. Suter TM, et al. Among authors: krushinski jh. Eur J Pharmacol. 2010 Dec 15;649(1-3):44-50. doi: 10.1016/j.ejphar.2010.08.055. Epub 2010 Sep 17. Eur J Pharmacol. 2010. PMID: 20851117

10

Characterization of type I 5 alpha-reductase activity in DU145 human prostatic adenocarcinoma cells.

Kaefer M, Audia JE, Bruchovsky N, Goode RL, Hsiao KC, Leibovitch IY, Krushinski JH, Lee C, Steidle CP, Sutkowski DM, Neubauer BL. Kaefer M, et al. Among authors: krushinski jh. J Steroid Biochem Mol Biol. 1996 May;58(2):195-205. doi: 10.1016/0960-0760(96)00020-9. J Steroid Biochem Mol Biol. 1996. PMID: 8809201

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