Functional interaction between retinoblastoma protein and stress-activated protein kinase in multiple myeloma cells

Cancer Res. 1999 Mar 15;59(6):1192-5.

Abstract

Previous studies have demonstrated that gamma-irradiation (IR)-induced apoptosis in multiple myeloma (MM) is associated with activation of stress-activated protein kinase (SAPK). In the present study, we examined the molecules downstream of SAPK/C-Jun N-terminal kinase (JNK), focusing on the role of retinoblastoma protein (Rb) during IR-induced MM cell apoptosis. The results demonstrate that IR activates SAPK/JNK, which associates with Rb both in vivo and in vitro. Far Western blot analysis confirms that SAPK/JNK binds directly to Rb. IR-activated SAPK/JNK phosphorylates Rb, and deletion of the phosphorylation site in the COOH terminus domain of Rb abrogates phosphorylation of Rb by SAPK/JNK. Taken together, our results suggest that Rb is a target protein of SAPK/JNK and that the association of SAPK/JNK and Rb mediates IR-induced apoptosis in MM cells.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Apoptosis / radiation effects
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
  • Enzyme Activation / radiation effects
  • Gamma Rays
  • Humans
  • JNK Mitogen-Activated Protein Kinases
  • Mitogen-Activated Protein Kinases*
  • Multiple Myeloma / enzymology
  • Multiple Myeloma / metabolism*
  • Phosphorylation / radiation effects
  • Protein Binding
  • Retinoblastoma Protein / metabolism*
  • Signal Transduction / physiology
  • Tumor Cells, Cultured

Substances

  • Retinoblastoma Protein
  • Calcium-Calmodulin-Dependent Protein Kinases
  • JNK Mitogen-Activated Protein Kinases
  • Mitogen-Activated Protein Kinases