Relationship between intracellular calcium-dependent process and protein-tyrosine phosphorylation in human platelets: studies of platelets from a patient with defective A23187-induced platelet aggregation

Clin Lab Haematol. 1999 Feb;21(1):29-32. doi: 10.1046/j.1365-2257.1999.00176.x.

Abstract

We had postulated that in a patient with defective calcium ionophore (A23187)-induced platelet aggregation, whose platelets showed normal intracellular Ca2+ mobilization in either the presence or absence of extracellular Ca2+ in response to A23187. A defect was present in an intracellular calcium-dependent process. We have now investigated whether the agonist-induced protein-tyrosine phosphorylation (PTP) was altered. Protein-tyrosine phosphorylation (PTP)-induced by A23187 in the patient's platelets was greatly diminished but that induced by thrombin was almost normal. These results suggest that an intracellular calcium-dependent process plays a fundamental role in A23187-induced PTP, whereas it does not in thrombin-induced PTP.

MeSH terms

  • Blood Platelet Disorders / blood
  • Blood Platelets / chemistry
  • Blood Platelets / drug effects
  • Calcimycin / pharmacology
  • Calcium / blood*
  • Extracellular Space / chemistry
  • Humans
  • Phosphorylation
  • Platelet Aggregation / drug effects
  • Protein-Tyrosine Kinases / blood
  • Protein-Tyrosine Kinases / metabolism*
  • Thrombin / pharmacology
  • Thrombin / therapeutic use

Substances

  • Calcimycin
  • Protein-Tyrosine Kinases
  • Thrombin
  • Calcium