Central and peripheral administration of endothelin-1 induces an increase in blood pressure in conscious trout

Am J Physiol. 1999 Apr;276(4):R1010-7. doi: 10.1152/ajpregu.1999.276.4.R1010.

Abstract

The central and peripheral cardiovascular effects of endothelin (ET)-1 and ET-3 were investigated in conscious rainbow trout. Both intracerebroventricular and intra-arterial injections of ET-1 (6. 25-25 pmol) but not ET-3 (25 pmol) caused a dose-dependent increase in mean dorsal aortic blood pressure and a concomitant decrease in heart rate. The hypertensive effects induced by intra-arterial and intracerebroventricular injection of ET-1 were associated with a significant (P < 0.05) increase in systemic vascular resistance. Intracerebroventricular injection of ET-1 induced a twofold higher pressor response than that caused by intra-arterial injection of ET-1 and provoked a barostatic gain that was reduced by 2.5- to 3-fold compared with that calculated after intra-arterial administration of the peptide. The ET receptor antagonist bosentan significantly (P < 0.05) attenuated these responses regardless of the route of administration. Finally, intra-arterial injection of ET-1 did not significantly modify plasma cortisol level. The present data demonstrate that intracerebroventricular and intra-arterial administration of very low doses of ET-1 produces hypertension in conscious trout. The lack of effect of ET-3 indicates that the hemodynamic actions of ET-1 are mediated both centrally and peripherally through ETA receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antihypertensive Agents / pharmacology
  • Blood Pressure / drug effects*
  • Bosentan
  • Cardiac Output / drug effects
  • Cardiovascular System / drug effects
  • Endothelin Receptor Antagonists
  • Endothelin-1 / administration & dosage*
  • Endothelin-1 / pharmacology
  • Heart Rate / drug effects
  • Hydrocortisone / blood
  • Injections, Intra-Arterial
  • Injections, Intraventricular
  • Oncorhynchus mykiss / blood
  • Oncorhynchus mykiss / physiology*
  • Sulfonamides / pharmacology

Substances

  • Antihypertensive Agents
  • Endothelin Receptor Antagonists
  • Endothelin-1
  • Sulfonamides
  • Bosentan
  • Hydrocortisone