Tyrosine phosphorylation of p62(Dok) induced by cell adhesion and insulin: possible role in cell migration

EMBO J. 1999 Apr 1;18(7):1748-60. doi: 10.1093/emboj/18.7.1748.

Abstract

Dok, a 62-kDa Ras GTPase-activating protein (rasGAP)-associated phosphotyrosyl protein, is thought to act as a multiple docking protein downstream of receptor or non-receptor tyrosine kinases. Cell adhesion to extracellular matrix proteins induced marked tyrosine phosphorylation of Dok. This adhesion-dependent phosphorylation of Dok was mediated, at least in part, by Src family tyrosine kinases. The maximal insulin-induced tyrosine phosphorylation of Dok required a Src family kinase. A mutant Dok (DokDeltaPH) that lacked its pleckstrin homology domain failed to undergo tyrosine phosphorylation in response to cell adhesion or insulin. Furthermore, unlike the wild-type protein, DokDeltaPH did not localize to subcellular membrane components. Insulin promoted the association of tyrosine-phosphorylated Dok with the adapter protein NCK and rasGAP. In contrast, a mutant Dok (DokY361F), in which Tyr361 was replaced by phenylalanine, failed to bind NCK but partially retained the ability to bind rasGAP in response to insulin. Overexpression of wild-type Dok, but not that of DokDeltaPH or DokY361F, enhanced the cell migratory response to insulin without affecting insulin activation of mitogen-activated protein kinase. These results identify Dok as a signal transducer that potentially links, through its interaction with NCK or rasGAP, cell adhesion and insulin receptors to the machinery that controls cell motility.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing
  • Animals
  • Base Sequence
  • Binding Sites
  • CHO Cells
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism
  • Cell Adhesion / physiology*
  • Cell Movement / physiology*
  • Cricetinae
  • DNA Primers / genetics
  • DNA-Binding Proteins*
  • Enzyme Activation / drug effects
  • Gene Expression
  • Humans
  • Insulin / pharmacology*
  • Mice
  • Oncogene Proteins / metabolism
  • Phosphoproteins / chemistry
  • Phosphoproteins / genetics
  • Phosphoproteins / metabolism*
  • Phosphorylation
  • RNA-Binding Proteins*
  • Subcellular Fractions / metabolism
  • Tyrosine / metabolism
  • src-Family Kinases / metabolism

Substances

  • Adaptor Proteins, Signal Transducing
  • DNA Primers
  • DNA-Binding Proteins
  • DOK1 protein, human
  • Dok1 protein, mouse
  • GAP-associated protein p62
  • Insulin
  • Nck protein
  • Oncogene Proteins
  • Phosphoproteins
  • RNA-Binding Proteins
  • Tyrosine
  • src-Family Kinases
  • Calcium-Calmodulin-Dependent Protein Kinases