Excretion and biotransformation of carboxymethyl-cysteine in rat, dog, monkey and man

Xenobiotica. 1978 Oct;8(10):621-8. doi: 10.3109/00498257809069574.

Abstract

1. Following an oral dose of S-carboxymethyl [35S]cysteine monkey (rhesus and African green), rat, dog, and man excreted 77,88,95, and 100% respectively of the 35S radioactivity in urine and 7.0, 2.5, 0.7, and 0.3% in faeces during a 3 to 4 day period. 2. The principal drug-related components excreted were unchanged carboxymethylcysteine, dicarboxymethyl sulphide and inorganic sulphate. 3. Rat, dog, and man excreted primarily dicarboxymethyl sulphide and unchanged carboxymethylcysteine and no inorganic sulphate (rat, 7%). 4. Monkey excreted largely inorganic sulphate, moderate amounts of dicarboxymethyl sulphide and a trace of unchanged drug.

MeSH terms

  • Animals
  • Biotransformation
  • Carbocysteine / blood
  • Carbocysteine / metabolism*
  • Carbocysteine / urine
  • Chromatography, High Pressure Liquid
  • Cysteine / analogs & derivatives*
  • Dogs
  • Feces / analysis
  • Female
  • Haplorhini
  • Humans
  • Macaca mulatta
  • Male
  • Rats
  • Species Specificity
  • Time Factors

Substances

  • Carbocysteine
  • Cysteine