Decreased striatal dopamine-receptor binding in sporadic ALS: glutamate hyperactivity?

Neurology. 1999 Apr 12;52(6):1275-7. doi: 10.1212/wnl.52.6.1275.

Abstract

The pathogenesis of ALS may be related to increased glutamatergic excitotoxicity. The striatum receives massive glutamatergic input. Animal studies suggest that glutamate decreases striatal D2-receptor synthesis. In drug-naive, sporadic ALS patients we demonstrated decreased striatal D2-receptor binding in vivo that could be partially reversed by the glutamatergic transmission blocker riluzole. Our findings support the glutamatergic excitotoxicity hypothesis in sporadic ALS.

MeSH terms

  • Aged
  • Amyotrophic Lateral Sclerosis / metabolism*
  • Corpus Striatum / metabolism*
  • Humans
  • Middle Aged
  • Pilot Projects
  • Receptors, Dopamine D2 / drug effects
  • Receptors, Dopamine D2 / metabolism*
  • Riluzole / pharmacology*

Substances

  • Receptors, Dopamine D2
  • Riluzole