Fra-1: a novel target for retinoid action

FEBS Lett. 1999 Apr 1;448(1):45-8. doi: 10.1016/s0014-5793(99)00326-9.

Abstract

Using a cDNA gene expression array system, we identified fra-1 as a novel target molecule for retinoid action in the human pancreatic carcinoma cell line Dan-G. Retinoid treatment resulted in a significant and time-dependent induction of the fra-1 expression on the post-transcriptional level. Supershift assays revealed that fra-1 participates in the activator protein 1 complex together with c-fos, c-jun and junB. Transient transfection experiments using a reporter plasmid containing an activator protein site upstream of the CAT reporter gene revealed that the phorbolester-induced CAT activity was suppressed by retinoids. Since fra-1 lacks a transactivation function, we therefore suggest that the retinoid-mediated induction of fra-1 might function as a negative regulator of the activator protein 1 activity in human pancreatic carcinoma cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Gene Expression Regulation / drug effects
  • Humans
  • Proto-Oncogene Proteins c-fos / genetics*
  • Retinoids / metabolism*
  • Retinoids / pharmacology
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transcription Factor AP-1 / metabolism
  • Tretinoin / metabolism
  • Tretinoin / pharmacology
  • Tumor Cells, Cultured

Substances

  • Proto-Oncogene Proteins c-fos
  • Retinoids
  • Transcription Factor AP-1
  • fos-related antigen 1
  • Tretinoin
  • Tetradecanoylphorbol Acetate