Dextran cross-linked gelatin microspheres as a drug delivery system

Eur J Pharm Biopharm. 1999 Mar;47(2):153-60. doi: 10.1016/s0939-6411(98)00076-9.

Abstract

This paper describes the use of oxidized dextran as a cross-linker for the preparation of gelatin microspheres. Microspheres were obtained by a thermal gelation method and their dissolution kinetic was examined. In order to find evidence of sugar mediated cross-linking, swelling tests and gelatin microspheres dissolution experiments were performed. The obtained results indicated that oxidized dextran can form a cross-linked gelatin network which can reduce the dissolution of gelatin. More interestingly, gelatin microspheres treated by both native and oxidized dextran slow down, even if to a different extent, the release of the antitumor drug TAPP-Br used as a model compound. Taken together, our results suggest that oxidized dextran could be an interesting means to cross-link gelatin microspheres allowing the use of this delivery formulation for controlled release of drugs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Dextrans / administration & dosage*
  • Drug Delivery Systems*
  • Gelatin / administration & dosage*
  • Microspheres

Substances

  • Dextrans
  • Gelatin