Molecular analysis of a new splice variant of the human melanocortin-1 receptor

FEBS Lett. 1999 May 21;451(2):137-41. doi: 10.1016/s0014-5793(99)00525-6.

Abstract

The primary hormonal regulator of pigmentation is melanocyte stimulating hormone derived from proopiomelanocortin by proteolytic processing. The melanocortin-1 receptor serves a key role in the regulation of pigmentation. We describe the identification of the first intron within a melanocortin receptor. A new melanocortin-1 receptor isoform, generated by alternative mRNA splicing, encodes an additional 65 amino acids at the predicted intracellular, C-terminal tail of the melanocortin-1 receptor. When expressed in heterologous cells, the new spliced form of the melanocortin-1 receptor (melanocortin-1 receptor B) appears pharmacologically similar to the non-spliced melanocortin-1 receptor. Melanocortin-1 receptor B is expressed in testis, fetal heart and melanomas.

MeSH terms

  • Alternative Splicing*
  • Amino Acid Sequence
  • Animals
  • Base Sequence
  • CHO Cells
  • Cloning, Molecular
  • Cricetinae
  • Expressed Sequence Tags
  • Humans
  • Inhibitory Concentration 50
  • Models, Genetic
  • Molecular Sequence Data
  • Polymorphism, Genetic
  • Protein Binding
  • Receptors, Corticotropin / genetics*
  • Receptors, Corticotropin / metabolism
  • Receptors, Melanocortin

Substances

  • Receptors, Corticotropin
  • Receptors, Melanocortin