Solution structure of core binding factor beta and map of the CBF alpha binding site

Nat Struct Biol. 1999 Jul;6(7):624-7. doi: 10.1038/10670.

Abstract

The core binding factor beta subunit (CBF beta) is the non-DNA binding subunit of the core-binding factors, transcription factors essential for multiple developmental processes including hematopoiesis and bone development. Chromosomal translocations involving the human CBFB gene are associated with a large percentage of human leukemias. The N-terminal 141 amino acids of CBF beta contains the heterodimerization domain for the DNA-binding CBF alpha subunits, and is sufficient for CBF beta function in vivo. Here we present the high-resolution solution structure of the CBF beta heterodimerization domain. It is a novel alpha/beta structure consisting of two three-stranded beta-sheets packed on one another in a sandwich arrangement, with four peripheral alpha-helices. The CBF alpha binding site on CBF beta has been mapped by chemical shift perturbation analysis.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Binding Sites
  • Circular Dichroism
  • Core Binding Factor alpha Subunits
  • Core Binding Factor beta Subunit
  • DNA-Binding Proteins / chemistry*
  • Humans
  • Magnetic Resonance Spectroscopy
  • Protein Structure, Secondary
  • Transcription Factor AP-2
  • Transcription Factors / chemistry*

Substances

  • CBFB protein, human
  • Core Binding Factor alpha Subunits
  • Core Binding Factor beta Subunit
  • DNA-Binding Proteins
  • Transcription Factor AP-2
  • Transcription Factors

Associated data

  • PDB/2JHB