A novel calcium signaling pathway targets the c-fos intragenic transcriptional pausing site

J Biol Chem. 1999 Oct 22;274(43):30439-46. doi: 10.1074/jbc.274.43.30439.

Abstract

In many cell types, increased intracellular calcium gives rise to a robust induction of c-fos gene expression. Here we show that in mouse Ltk(-) fibroblasts, calcium ionophore acts in synergy with either cAMP or PMA to strongly induce the endogenous c-fos gene. Run-on analysis shows that this corresponds to a substantial increase in active polymerases on downstream gene sequences, i.e. relief of an elongation block by calcium. Correspondingly a chimeric gene, in which the human metallothionein promoter is fused to the fos gene, is strongly induced by ionophore alone, unlike a c-fos promoter/beta-globin coding unit chimeric construct. Internal deletions in the hMT-fos reporter localize the intragenic calcium regulatory element to the 5' portion of intron 1, thereby confirming and extending previous in vitro mapping data. Ionophore induced cAMP response element-binding protein phosphorylation on Ser(133) without affecting the extracellular signal-regulated kinase cascade. Surprisingly, induction involved neither CaM-Ks nor calcineurin, while the calmodulin antagonist W7 activated c-fos transcription on its own. These data suggest that a novel calcium signaling pathway mediates intragenic regulation of c-fos expression via suppression of a transcriptional pause site.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 1-Methyl-3-isobutylxanthine / pharmacology
  • 5' Untranslated Regions / genetics
  • 8-Bromo Cyclic Adenosine Monophosphate / pharmacology
  • Animals
  • Calcimycin / pharmacology
  • Calcineurin / metabolism
  • Calcium / metabolism*
  • Calmodulin / antagonists & inhibitors
  • Cyclic AMP / physiology
  • Cyclic AMP Response Element-Binding Protein / metabolism
  • Gene Expression Regulation* / drug effects
  • Genes, Reporter
  • Genes, fos*
  • Humans
  • Introns
  • L Cells
  • Metallothionein / genetics
  • Mice
  • Mitogen-Activated Protein Kinases / metabolism
  • Phosphorylation
  • Promoter Regions, Genetic
  • Recombinant Fusion Proteins / biosynthesis
  • Serine
  • Signal Transduction / physiology*
  • Sulfonamides / pharmacology
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transcription, Genetic*

Substances

  • 5' Untranslated Regions
  • Calmodulin
  • Cyclic AMP Response Element-Binding Protein
  • Recombinant Fusion Proteins
  • Sulfonamides
  • 8-Bromo Cyclic Adenosine Monophosphate
  • Calcimycin
  • Serine
  • W 7
  • Metallothionein
  • Cyclic AMP
  • Mitogen-Activated Protein Kinases
  • Calcineurin
  • Tetradecanoylphorbol Acetate
  • Calcium
  • 1-Methyl-3-isobutylxanthine