Fish model for assessing the in vivo estrogenic potency of the mycotoxin zearalenone and its metabolites

Sci Total Environ. 1999 Sep 15;236(1-3):153-61. doi: 10.1016/s0048-9697(99)00275-2.

Abstract

The in vivo estrogenic potency of zearalenone (ZEA), a mycotoxin produced by different strains of Fusarium fungi, and its metabolites (alpha- and beta-zearalenol), have been studied in fish. Estrogenicity was evaluated using an in vitro competitive receptor binding assay and in vivo induction of vitellogenesis and zonagenesis, two estrogen receptor (ER)-mediated responses that are integral aspects of fish oogenesis. The ER binding affinities of alpha-zearalenol and ZEA in rainbow trout (Oncorhynchus mykiss) were approximately 1/150 and 1/300 to that of estradiol, respectively. Juvenile salmon (Salmo salar) were exposed to a single intraperitoneal injection of ZEA, alpha-zearalenol and beta-zearalenol (each at 1 and 10 mg/kg) and compared to fish injected with estradiol-17 beta (E2; 5 mg/kg) and controls. Using indirect enzyme-linked immunosorbent assay (ELISA) with homologous antibodies, a dose-dependent induction of vitellogenin (Vtg) and eggshell zona radiata proteins (Zr-proteins) were observed 7 days after exposure to ZEA and alpha-zearalenol. beta-Zearalenol did not elevate plasma Vtg levels, but a non-significant elevation of plasma Zr-proteins levels was observed at the highest dose (10 mg/kg). Generally, alpha-zearalenol and ZEA possess estrogenic potencies that are approximately 50% compared to that of E2, and their order of estrogenic potency (in both in vitro receptor competitive binding and in vivo induction of Vtg and Zr-proteins levels) is: alpha-zearalenol > ZEA > beta-zearalenol. Our results show that blood plasma analysis of Vtg and Zr-proteins levels provides a suitable in vivo fish model for assessing the estrogenic potencies of ZEA and its metabolites.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding, Competitive
  • Egg Proteins / biosynthesis
  • Estradiol / metabolism
  • Estradiol / pharmacology
  • Estrogens, Non-Steroidal / metabolism
  • Estrogens, Non-Steroidal / pharmacology*
  • Female
  • In Vitro Techniques
  • Male
  • Models, Biological
  • Oncorhynchus mykiss
  • Oogenesis / drug effects
  • Receptors, Estrogen / drug effects
  • Receptors, Estrogen / metabolism
  • Salmo salar
  • Vitellogenins / biosynthesis
  • Zearalenone / metabolism
  • Zearalenone / pharmacology*
  • Zeranol / analogs & derivatives
  • Zeranol / pharmacology

Substances

  • Egg Proteins
  • Estrogens, Non-Steroidal
  • Receptors, Estrogen
  • Vitellogenins
  • zearalenol
  • Estradiol
  • Zearalenone
  • Zeranol