L-type calcium channels and GSK-3 regulate the activity of NF-ATc4 in hippocampal neurons

Nature. 1999 Oct 14;401(6754):703-8. doi: 10.1038/44378.

Abstract

The molecular basis of learning and memory has been the object of several recent advances, which have focused attention on calcium-regulated pathways controlling transcription. One of the molecules implicated by pharmacological, biochemical and genetic approaches is the calcium/calmodulin-regulated phosphatase, calcineurin. In lymphocytes, calcineurin responds to specific calcium signals and regulates expression of several immediate early genes by controlling the nuclear import of the NF-ATc family of transcription factors. Here we show that NF-ATc4/NF-AT3 in hippocampal neurons can rapidly translocate from cytoplasm to nucleus and activate NF-AT-dependent transcription in response to electrical activity or potassium depolarization. The calcineurin-mediated translocation is critically dependent on calcium entry through L-type voltage-gated calcium channels. GSK-3 can phosphorylate NF-ATc4, promoting its export from the nucleus and antagonizing NF-ATc4-dependent transcription. Furthermore, we show that induction of the inositol 1,4,5-trisphosphate receptor type 1 is controlled by the calcium/calcineurin/NF-ATc pathway. This provides a new perspective on the function of calcineurin in the central nervous system and indicates that NF-AT-mediated gene expression may be involved in the induction of hippocampal synaptic plasticity and memory formation.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Biological Transport
  • Calcineurin / metabolism
  • Calcium / metabolism
  • Calcium Channels / metabolism
  • Calcium Channels, L-Type / metabolism*
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
  • Cell Nucleus / metabolism
  • Cells, Cultured
  • Cytoplasm / metabolism
  • DNA-Binding Proteins / metabolism*
  • Electrophysiology
  • Gene Expression Regulation
  • Glycogen Synthase Kinase 3
  • Green Fluorescent Proteins
  • Hippocampus / cytology
  • Hippocampus / metabolism*
  • Inositol 1,4,5-Trisphosphate Receptors
  • Luminescent Proteins / genetics
  • NFATC Transcription Factors
  • Neurons / metabolism*
  • Nuclear Proteins*
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Transcription Factors / metabolism*
  • Transcription, Genetic

Substances

  • Calcium Channels
  • Calcium Channels, L-Type
  • DNA-Binding Proteins
  • Inositol 1,4,5-Trisphosphate Receptors
  • Luminescent Proteins
  • NFATC Transcription Factors
  • Nuclear Proteins
  • Receptors, Cytoplasmic and Nuclear
  • Transcription Factors
  • Green Fluorescent Proteins
  • Calcium-Calmodulin-Dependent Protein Kinases
  • Glycogen Synthase Kinase 3
  • Calcineurin
  • Calcium