The nucleotide-binding site of the sarcoplasmic reticulum Ca-ATPase is conformationally altered in aged skeletal muscle

Biochemistry. 1999 Nov 9;38(45):14887-96. doi: 10.1021/bi991125n.

Abstract

Cellular conditions in senescent skeletal muscle have been shown to result in the loss of conformational stability of the sarcoplasmic reticulum (SR) Ca-ATPase. To identify underlying structural features of age-modified Ca-ATPase, we have utilized the fluorescence properties of protein-bound probes to assess both local and global structure. We find conformational changes that include an age-related decrease in the apparent binding affinity to high affinity calcium sites detected by fluorescence signals in both tryptophans within nearby membrane-spanning helices and fluorescein isothiocyanate (FITC) bound distally to Lys(515) within the nucleotide-binding site. In addition, a substantial (80%) age-related increase in the accessibility to soluble quenchers of fluorescence of FITC is observed without concomitant changes in bimolecular quenching constants (k(q)) for protein-bound IAEDANS, also within the nucleotide-binding domain, and tryptophans within the membrane. Using fluorescence resonance energy transfer to measure distances between IAEDANS and FITC across the nucleotide-binding domain, we find no significant age-related change in the mean donor-acceptor distance; however, significant increases are observed in the conformational heterogeneity of this domain, as assessed by the width at half-maximum (HW) of the distance distribution, increasing with age from 29.4 +/- 0.8 A to 42.5 +/- 1. 1 A. Circular dichroism indicates that the average secondary structure is unaltered with age. Thus, these data suggest tertiary structural alterations in specific regions around the nucleotide-binding site rather than global conformational changes.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aging*
  • Animals
  • Binding Sites
  • Calcium-Transporting ATPases / metabolism*
  • Circular Dichroism
  • Energy Transfer
  • Fluorescein-5-isothiocyanate
  • Fluorescent Dyes / metabolism
  • Models, Biological
  • Muscle, Skeletal / enzymology*
  • Muscle, Skeletal / metabolism
  • Naphthalenesulfonates / metabolism
  • Nucleotides / metabolism*
  • Protein Conformation
  • Protein Structure, Secondary
  • Rats
  • Rats, Inbred F344
  • Sarcoplasmic Reticulum / enzymology*
  • Solvents
  • Spectrometry, Fluorescence

Substances

  • Fluorescent Dyes
  • Naphthalenesulfonates
  • Nucleotides
  • Solvents
  • 1,5-I-AEDANS
  • Calcium-Transporting ATPases
  • Fluorescein-5-isothiocyanate