Protective effect of 3-aminobenzamide, an inhibitor of poly (ADP-ribose) synthetase, against laryngeal injury in rats

Am J Respir Crit Care Med. 1999 Nov;160(5 Pt 1):1743-9. doi: 10.1164/ajrccm.160.5.9902024.

Abstract

The effect of 3-aminobenzamide, an inhibitor of poly (ADP-ribose) synthetase activity, was evaluated in a rat model of laryngeal injury induced by endotracheal intubation for 1 h. At 1 h after extubation, the laryngeal damage was characterized by areas of mucosal necrosis, submucosal edema, swelling of subglottic glands, and submucosal infiltration of inflammatory cells. Activity of myeloperoxidase, a marker of neutrophil infiltration, was also markedly increased into the damaged tissue. Immunohistochemistry for nitrotyrosine, an index of nitrosative stress, showed an intense staining in the inflamed larynx. Treatment with 3-aminobenzamide (10 mg/kg intraperitoneally) significantly reduced the appearance of mucosal damage and was associated with a significant reduction of tissue myeloperoxidase activity and nitrotyrosine immunoreactivity in the larynx. The results of this study suggest that poly (ADP-ribose) synthetase may play a role in the inflammatory process after laryngeal intubation and extubation, and administration of 3-aminobenzamide may be a beneficial therapeutic approach.

MeSH terms

  • Animals
  • Benzamides / pharmacology*
  • Enzyme Inhibitors / pharmacology*
  • Immunohistochemistry
  • Intubation, Intratracheal / adverse effects*
  • Laryngeal Mucosa / chemistry
  • Laryngeal Mucosa / pathology
  • Larynx / injuries*
  • Larynx / pathology
  • Male
  • Neutrophils / pathology
  • Peroxidase / analysis
  • Poly(ADP-ribose) Polymerase Inhibitors*
  • Rats
  • Rats, Wistar
  • Tyrosine / analogs & derivatives
  • Tyrosine / analysis
  • Wounds and Injuries / etiology
  • Wounds and Injuries / pathology

Substances

  • Benzamides
  • Enzyme Inhibitors
  • Poly(ADP-ribose) Polymerase Inhibitors
  • 3-nitrotyrosine
  • Tyrosine
  • 3-aminobenzamide
  • Peroxidase