5-HT1A autoreceptor desensitization by chronic ultramild stress in mice

Neuroreport. 1999 Nov 8;10(16):3369-74. doi: 10.1097/00001756-199911080-00021.

Abstract

Electrophysiological and biochemical approaches were used to assess possible changes in central 5-HT neurotransmission in mice that had been subjected to chronic ultramild stress for 8 weeks. This treatment produced a significant decrease in the potency of the 5-HT1A agonist ipsapirone to inhibit the electrical activity of serotoninergic neurons in the dorsal raphe nucleus, without modifying 5-HT1A receptor binding in various brain areas. These data demonstrate that chronic ultramild stress triggers a long term and durable functional desensitization of somatodendritic 5-HT1A autoreceptors in mice.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / physiology
  • Animals
  • Brain Chemistry / physiology
  • Chronic Disease
  • Corticosterone / metabolism
  • Electrophysiology
  • Hydroxyindoleacetic Acid / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred DBA
  • Neurons / metabolism
  • Neurons / physiology
  • Pyrimidines / pharmacology
  • Receptors, Serotonin / drug effects
  • Receptors, Serotonin / physiology*
  • Receptors, Serotonin, 5-HT1
  • Serotonin / metabolism
  • Serotonin / physiology
  • Serotonin Receptor Agonists / pharmacology
  • Stress, Psychological / physiopathology*
  • Synaptic Transmission / physiology

Substances

  • Pyrimidines
  • Receptors, Serotonin
  • Receptors, Serotonin, 5-HT1
  • Serotonin Receptor Agonists
  • Serotonin
  • Hydroxyindoleacetic Acid
  • ipsapirone
  • Corticosterone