Porous balloon delivery of S-dC28 does not prevent restenosis in the porcine coronary artery model of balloon injury

Antisense Nucleic Acid Drug Dev. 1999 Dec;9(6):549-53. doi: 10.1089/oli.1.1999.9.549.

Abstract

Phosphorothioate (PS) oligodeoxynucleotides (ODN) inhibit vascular smooth muscle cell proliferation through antisense and G-quartet aptameric mechanisms. PS-ODN such as the cytidine homopolymers, have been demonstrated to have non-G-quartet, nonsequence-specific inhibitory effects in a rat carotid balloon injury model of neointimal proliferation. We sought to test the efficacy of S-dC28, a cytidine homopolymer lacking G-quartets, on neointimal proliferation in the porcine coronary artery model of balloon injury. A total of 23 animals (11 controls, 12 treated) were subjected to balloon injury in a coronary artery, followed by infusion of control solution or S-dC28 via porous balloon, the Scimed Dispatch Coronary Infusion Catheter. After a mean interval of 49 days, the animals were killed, and the target coronary segments were examined histologically. S-dC28 did not significantly inhibit neointimal formation. Fluorescein isothiocyanate (FITC)-labeled S-dC28 was present in the intima and media immediately after administration but was present mainly within the adventitia 3 hours after administration. S-dC28, when delivered by a Scimed Dispatch Coronary Infusion Catheter (Maple Grove, MN), did not significantly affect neointimal proliferation after balloon injury in a porcine coronary artery model.

Publication types

  • Letter
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angioplasty, Balloon, Coronary / adverse effects
  • Animals
  • Cell Division
  • Coronary Vessels / drug effects
  • Coronary Vessels / injuries*
  • Coronary Vessels / pathology
  • Disease Models, Animal
  • Fluorescein-5-isothiocyanate
  • Fluorescent Dyes
  • Muscle, Smooth, Vascular / pathology
  • Oligodeoxyribonucleotides / administration & dosage*
  • Oligodeoxyribonucleotides / genetics
  • Rats
  • Swine
  • Thionucleotides / administration & dosage
  • Thionucleotides / genetics

Substances

  • Fluorescent Dyes
  • Oligodeoxyribonucleotides
  • Thionucleotides
  • Fluorescein-5-isothiocyanate