Calcineurin is downstream of the inositol 1,4,5-trisphosphate receptor in the apoptotic and cell growth pathways

J Biol Chem. 2000 Mar 3;275(9):6417-20. doi: 10.1074/jbc.275.9.6417.

Abstract

The inositol 1,4,5-trisphosphate receptor (IP(3)R) is a calcium (Ca(2+)) release channel found on the endoplasmic reticulum of virtually all types of cells. Human T lymphocytes (Jurkat) that are made deficient in IP(3)R do not generate Ca(2+) signals in response to T cell receptor stimulation, fail to translocate the nuclear factor for activated T cells to the nucleus, and are remarkably resistant to induction of apoptosis with CD95 (Fas), dexamethasone, gamma irradiation, and T cell receptor stimulation using anti-CD3 antibody. Expression of constitutively active calcineurin A in IP(3)R-deficient T cells restored nuclear factor for activated T cells translocation to the nucleus and dephosphorylation of Bad and rendered the cells sensitive to apoptotic inducers. Induction of apoptosis required both active calcineurin A (DeltaCnA) and activation-dependent colocalization of CnA with its substrate. Thus, the Ca(2+)-dependent phosphatase calcineurin (CnA) is downstream of the IP(3)R in both the cell growth and apoptotic signaling pathways.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Apoptosis*
  • CD3 Complex / metabolism
  • Calcineurin / genetics
  • Calcineurin / metabolism*
  • Calcium / metabolism
  • Calcium Channels / deficiency*
  • Carrier Proteins / metabolism
  • Cell Division*
  • DNA-Binding Proteins / metabolism
  • Green Fluorescent Proteins
  • Humans
  • Inositol 1,4,5-Trisphosphate Receptors
  • Luminescent Proteins
  • Microscopy, Fluorescence
  • NFATC Transcription Factors
  • Nuclear Proteins / metabolism
  • Phosphorylation
  • Receptors, Cytoplasmic and Nuclear / deficiency*
  • Signal Transduction*
  • T-Lymphocytes
  • Transcription Factors / metabolism
  • Transfection
  • bcl-Associated Death Protein

Substances

  • BAD protein, human
  • CD3 Complex
  • Calcium Channels
  • Carrier Proteins
  • DNA-Binding Proteins
  • ITPR1 protein, human
  • Inositol 1,4,5-Trisphosphate Receptors
  • Luminescent Proteins
  • NFATC Transcription Factors
  • Nuclear Proteins
  • Receptors, Cytoplasmic and Nuclear
  • Transcription Factors
  • bcl-Associated Death Protein
  • Green Fluorescent Proteins
  • Calcineurin
  • Calcium