The heparin-binding site in tetranectin is located in the N-terminal region and binding does not involve the carbohydrate recognition domain

Biochem J. 2000 Apr 1;347 Pt 1(Pt 1):83-7.

Abstract

Tetranectin is a homotrimeric plasma and extracellular-matrix protein that binds plasminogen and complex sulphated polysaccharides including heparin. In terms of primary and tertiary structure, tetranectin is related to the collectin family of Ca(2+)-binding C-type lectins. Tetranectin is encoded in three exons. Exon 3 encodes the carbohydrate recognition domain, which binds to kringle 4 in plasminogen at low levels of Ca(2+). Exon 2 encodes an alpha-helix, which is necessary and sufficient to govern the trimerization of tetranectin by assembling into a triple-helical coiled-coil structural element. Here we show that the heparin-binding site in tetranectin resides not in the carbohydrate recognition domain but within the N-terminal region, comprising the 16 amino acid residues encoded by exon 1. In particular, the lysine residues in the decapeptide segment KPKKIVNAKK (tetranectin residues 6-15) are shown to be of primary importance in heparin binding.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Amino Acid Substitution
  • Animals
  • Base Sequence
  • Binding Sites
  • Blood Proteins / chemistry*
  • Blood Proteins / genetics
  • Blood Proteins / metabolism*
  • Calcium / metabolism
  • Chromatography, Affinity
  • Exons
  • Heparin / metabolism*
  • Humans
  • Kinetics
  • Lectins / chemistry
  • Lectins / metabolism
  • Lectins, C-Type*
  • Mice
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Plasminogen / chemistry
  • Plasminogen / metabolism
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Sequence Alignment
  • Sequence Homology, Amino Acid

Substances

  • Blood Proteins
  • Lectins
  • Lectins, C-Type
  • Recombinant Proteins
  • tetranectin
  • Plasminogen
  • Heparin
  • Calcium