Abstract
Epsin (Eps15 interactor) is a cytosolic protein involved in clathrin-mediated endocytosis via its direct interactions with clathrin, the clathrin adaptor AP-2, and Eps15. The NH(2)-terminal portion of epsin contains a phylogenetically conserved module of unknown function, known as the ENTH domain (epsin NH(2)-terminal homology domain). We have now solved the crystal structure of rat epsin 1 ENTH domain to 1.8 A resolution. This domain is structurally similar to armadillo and Heat repeats of beta-catenin and karyopherin-beta, respectively. We have also identified and characterized the interaction of epsin 1, via the ENTH domain, with the transcription factor promyelocytic leukemia Zn(2)+ finger protein (PLZF). Leptomycin B, an antifungal antibiotic, which inhibits the Crm1- dependent nuclear export pathway, induces an accumulation of epsin 1 in the nucleus. These findings suggest that epsin 1 may function in a signaling pathway connecting the endocytic machinery to the regulation of nuclear function.
Publication types
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Research Support, Non-U.S. Gov't
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Research Support, U.S. Gov't, P.H.S.
MeSH terms
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Adaptor Proteins, Vesicular Transport
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Amino Acid Sequence
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Animals
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Armadillo Domain Proteins
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Calcium-Binding Proteins / metabolism*
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Carrier Proteins / chemistry*
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Carrier Proteins / metabolism
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Cell Line
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Cell Nucleus / metabolism
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Crystallography, X-Ray
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Cytoskeletal Proteins / chemistry
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Cytosol / metabolism
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DNA-Binding Proteins / metabolism*
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Drosophila Proteins*
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Fluorescent Antibody Technique
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Insect Proteins / chemistry
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Models, Molecular
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Molecular Sequence Data
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Neuropeptides / chemistry*
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Neuropeptides / metabolism
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Phosphoproteins / metabolism*
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Protein Binding
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Rats
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Sequence Alignment
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Trans-Activators*
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Transcription Factors / metabolism*
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Vesicular Transport Proteins*
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Zinc Fingers
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beta Catenin
Substances
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Adaptor Proteins, Vesicular Transport
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Armadillo Domain Proteins
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Calcium-Binding Proteins
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Carrier Proteins
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Ctnnb1 protein, rat
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Cytoskeletal Proteins
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DNA-Binding Proteins
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Drosophila Proteins
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Insect Proteins
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Neuropeptides
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Phosphoproteins
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Trans-Activators
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Transcription Factors
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Vesicular Transport Proteins
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beta Catenin
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epsin