Structure-function relationships in yeast tubulins

Mol Biol Cell. 2000 May;11(5):1887-903. doi: 10.1091/mbc.11.5.1887.

Abstract

A comprehensive set of clustered charged-to-alanine mutations was generated that systematically alter TUB1, the major alpha-tubulin gene of Saccharomyces cerevisiae. A variety of phenotypes were observed, including supersensitivity and resistance to the microtubule-destabilizing drug benomyl, lethality, and cold- and temperature-sensitive lethality. Many of the most benomyl-sensitive tub1 alleles were synthetically lethal in combination with tub3Delta, supporting the idea that benomyl supersensitivity is a rough measure of microtubule instability and/or insufficiency in the amount of alpha-tubulin. The systematic tub1 mutations were placed, along with the comparable set of tub2 mutations previously described, onto a model of the yeast alpha-beta-tubulin dimer based on the three-dimensional structure of bovine tubulin. The modeling revealed a potential site for binding of benomyl in the core of beta-tubulin. Residues whose mutation causes cold sensitivity were concentrated at the lateral and longitudinal interfaces between adjacent subunits. Residues that affect binding of the microtubule-binding protein Bim1p form a large patch across the exterior-facing surface of alpha-tubulin in the model. Finally, the positions of the mutations suggest that proximity to the alpha-beta interface may account for the finding of synthetic lethality of five viable tub1 alleles with the benomyl-resistant but otherwise entirely viable tub2-201 allele.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Benomyl / metabolism
  • Binding Sites
  • Cattle
  • Cell Cycle Proteins / metabolism
  • Cold Temperature
  • Fungal Proteins / chemistry*
  • Fungal Proteins / genetics
  • Fungal Proteins / metabolism*
  • Microtubule Proteins / metabolism
  • Microtubules / metabolism
  • Models, Molecular
  • Multigene Family
  • Mutation
  • Phenotype
  • Protein Conformation
  • Saccharomyces cerevisiae / metabolism*
  • Saccharomyces cerevisiae / physiology
  • Saccharomyces cerevisiae Proteins*
  • Structure-Activity Relationship
  • Tubulin / chemistry*
  • Tubulin / genetics
  • Tubulin / metabolism*

Substances

  • BIM1 protein, S cerevisiae
  • Cell Cycle Proteins
  • Fungal Proteins
  • Microtubule Proteins
  • Saccharomyces cerevisiae Proteins
  • Tubulin
  • Benomyl