Matrix mini-tablets based on starch/microcrystalline wax mixtures

Int J Pharm. 2000 Apr 20;199(2):195-203. doi: 10.1016/s0378-5173(00)00383-5.

Abstract

Matrix mini-tablets based on a combination of microcrystalline waxes and starch derivatives were prepared using ibuprofen as a model drug. The production of mini-tablets was preferred over the production of pellets, as up-scaling of the pelletisation process seemed problematic. Prior to tabletting, melt granulation in a hot stage screw extruder and milling were required. The in vitro drug release was varied using microcrystalline waxes with a different melting range, the slowest drug release being obtained with a formulation containing a microcrystalline wax with a melting range between 68 and 72 degrees C. Generally speaking increasing the wax concentration resulted in a slower drug release. In vitro drug release profiles were also modified using different starches and mixtures of starches. Increasing the ibuprofen concentration to 70% resulted in a faster drug release rate.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Capsules*
  • Chemistry, Pharmaceutical / methods*
  • Delayed-Action Preparations
  • Ibuprofen / administration & dosage
  • Microspheres
  • Starch*
  • Waxes*
  • X-Ray Diffraction

Substances

  • Capsules
  • Delayed-Action Preparations
  • Waxes
  • Starch
  • Ibuprofen