Mechanism of kappa B DNA binding by Rel/NF-kappa B dimers

J Biol Chem. 2000 Aug 11;275(32):24392-9. doi: 10.1074/jbc.M003784200.

Abstract

The DNA binding of three different NF-kappaB dimers, the p50 and p65 homodimers and the p50/p65 heterodimer, has been examined using a combination of gel mobility shift and fluorescence anisotropy assays. The NF-kappaB p50/p65 heterodimer is shown here to bind the kappaB DNA target site of the immunoglobulin kappa enhancer (Ig-kappaB) with an affinity of approximately 10 nm. The p50 and p65 homodimers bind to the same site with roughly 5- and 15-fold lower affinity, respectively. The nature of the binding isotherms indicates a cooperative mode of binding for all three dimers to the DNA targets. We have further characterized the role of pH, salt, and temperature on the formation of the p50/p65 heterodimer-Ig-kappaB complex. The heterodimer binds to the Ig-kappaB DNA target in a pH-dependent manner, with the highest affinity between pH 7.0 and 7.5. A strong salt-dependent interaction between Ig-kappaB and the p50/p65 heterodimer is observed, with optimum binding occurring at monovalent salt concentrations below 75 mm, with binding becoming virtually nonspecific at a salt concentration of 200 mm. Binding of the heterodimer to DNA was unchanged across a temperature range between 4 degrees C and 42 degrees C. The sensitivity to ionic environment and insensitivity to temperature indicate that NF-kappaB p50/p65 heterodimers form complexes with specific DNA in an entropically driven manner.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Substitution
  • Binding Sites
  • DNA / chemistry*
  • DNA / metabolism*
  • Dimerization
  • HIV Long Terminal Repeat
  • Hydrogen-Ion Concentration
  • Kinetics
  • Models, Chemical
  • Mutagenesis, Site-Directed
  • NF-kappa B / chemistry*
  • NF-kappa B / metabolism*
  • Oligodeoxyribonucleotides / chemistry
  • Oligodeoxyribonucleotides / metabolism*
  • Protein Multimerization
  • Proto-Oncogene Proteins c-rel / chemistry*
  • Proto-Oncogene Proteins c-rel / metabolism*
  • Thermodynamics

Substances

  • NF-kappa B
  • Oligodeoxyribonucleotides
  • Proto-Oncogene Proteins c-rel
  • DNA