Regulation of the hTERT telomerase catalytic subunit by the c-Abl tyrosine kinase

Curr Biol. 2000 May 18;10(10):568-75. doi: 10.1016/s0960-9822(00)00483-8.

Abstract

Background: Telomeres consist of repetitive (TTAGGG) DNA sequences that are maintained by the multisubunit telomerase ribonucleoprotein. Telomerase consists of an RNA, which serves as template for the sequence tracts, and a catalytic subunit that functions in reverse transcription of the RNA template. Cloning and characterization of the human catalytic subunit of telomerase (hTERT) has supported a role in cell transformation. How telomerase activity is regulated, however, is largely unknown.

Results: We show here that hTERT associates directly with the c-Abl protein tyrosine kinase. We also found that c-Abl phosphorylates hTERT and inhibits hTERT activity. Moreover, our findings demonstrate that exposure of cells to ionizing radiation induces tyrosine phosphorylation of hTERT by a c-Abl-dependent mechanism. The functional significance of the c-Abl-hTERT interaction is supported by the demonstration that cells deficient in c-Abl show telomere lengthening.

Conclusions: The ubiquitously expressed c-Abl tyrosine kinase is activated by DNA double-strand breaks. Our finding of telomere lengthening in c-Abl-deficient cells and the functional interactions between c-Abl and hTERT support a role for c-Abl in the regulation of telomerase function.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Catalytic Domain
  • Cells, Cultured
  • DNA-Binding Proteins
  • Fibroblasts
  • Gene Expression Regulation, Enzymologic*
  • Humans
  • Immunoblotting
  • Phosphorylation
  • Precipitin Tests
  • Proto-Oncogene Proteins c-abl / genetics
  • Proto-Oncogene Proteins c-abl / metabolism*
  • RNA*
  • Telomerase / genetics*
  • Telomerase / metabolism*
  • Telomere / physiology
  • Transfection

Substances

  • DNA-Binding Proteins
  • telomerase RNA
  • RNA
  • Proto-Oncogene Proteins c-abl
  • Telomerase