New quinolinic derivatives as centrally active antioxidants

Bioorg Med Chem Lett. 2000 May 1;10(9):935-9. doi: 10.1016/s0960-894x(00)00122-0.

Abstract

A series of new 1,2-dihydro and 1,2,3,4-tetrahydroquinolines, synthesized from the corresponding propargylaniline intermediates, have been developed as antioxidants for the potential treatment of pathologies implicating central oxidative stress.

MeSH terms

  • Animals
  • Antioxidants / chemical synthesis*
  • Antioxidants / pharmacology*
  • Cell Line
  • Electrons
  • Ethoxyquin / chemistry
  • Hippocampus / cytology
  • Hippocampus / drug effects
  • Hippocampus / metabolism
  • Isoquinolines / chemistry
  • Isoquinolines / pharmacology
  • Mice
  • Neurons / drug effects
  • Neuroprotective Agents / chemical synthesis
  • Neuroprotective Agents / pharmacology
  • Oxidants / toxicity
  • Oxidative Stress / drug effects
  • Quinolinic Acids / chemical synthesis*
  • Quinolinic Acids / pharmacology*
  • Structure-Activity Relationship
  • Vitamin E / pharmacology
  • tert-Butylhydroperoxide / antagonists & inhibitors
  • tert-Butylhydroperoxide / toxicity

Substances

  • Antioxidants
  • Isoquinolines
  • Neuroprotective Agents
  • Oxidants
  • Quinolinic Acids
  • Vitamin E
  • tert-Butylhydroperoxide
  • Ethoxyquin