Effects of fedotozine on gastric emptying and upper gastrointestinal symptoms in diabetic gastroparesis

Aliment Pharmacol Ther. 2000 Jul;14(7):937-43. doi: 10.1046/j.1365-2036.2000.00790.x.

Abstract

Background: Delayed gastric emptying and upper gastrointestinal symptoms occur frequently in patients with diabetes mellitus.

Aim: To evaluate the effects of fedotozine on gastric emptying and gastrointestinal symptoms in diabetic gastroparesis.

Methods: Thirty-one diabetic patients (20 type 1, 11 type 2) with gastroparesis were randomized to receive fedotozine (30 mg as the tartrate) or placebo t.d.s. Measurements of gastric emptying (100 g ground beef labelled with 20 MBq 99mTc-sulphur colloid chicken liver and 150 mL 10% dextrose labelled with 10 MBq 113mIn-DTPA) and gastrointestinal symptoms were performed before and after 12-16 days of treatment. Data are the mean +/- s.d.

Results: Of the 31 patients enrolled, two were excluded from analysis. Data from the remaining 29 patients (18 type 1, 11 type 2; 22 female, seven male), aged 42.7 +/- 11.1 years (of whom 14 were randomized to fedotozine and 15 to placebo), were analysed. Fedotozine had no effect on either gastric emptying (solid retention at 100 min; fedotozine: baseline, 84 +/- 15%; treatment, 73 +/- 23% vs. placebo: baseline, 83 +/- 10%; treatment, 70 +/- 20%) or liquid 50% emptying time (fedotozine: baseline, 59 +/- 32 min; treatment, 58 +/- 38 min vs. placebo: baseline, 44 +/- 9 min; treatment, 43 +/- 21 min) or gastrointestinal symptoms (fedotozine: baseline, 4.4 +/- 2.9; treatment, 4.1 +/- 3.9 vs. placebo: baseline, 4.9 +/- 4.2; treatment, 4.8 +/- 3.9).

Conclusions: Fedotozine has no effect on gastric emptying in patients with diabetic gastroparesis.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Anorexia / drug therapy
  • Anorexia / etiology
  • Benzyl Compounds / pharmacology
  • Benzyl Compounds / therapeutic use*
  • Blood Glucose / metabolism
  • Diabetes Complications
  • Female
  • Gastric Emptying / drug effects*
  • Gastroparesis / blood
  • Gastroparesis / drug therapy*
  • Gastroparesis / physiopathology
  • Heartburn / drug therapy
  • Heartburn / etiology
  • Humans
  • Male
  • Outcome Assessment, Health Care
  • Propylamines / pharmacology
  • Propylamines / therapeutic use*

Substances

  • Benzyl Compounds
  • Blood Glucose
  • Propylamines
  • fedotozine