Synthesis of glycosyl(thio)ureido sugars via carbodiimides and their conformational behaviour in water

Carbohydr Res. 2000 Jun 16;326(3):161-75. doi: 10.1016/s0008-6215(00)00040-9.

Abstract

The preparation of sugar ureas and thioureas by nucleophilic addition of water or hydrogen sulfide, respectively, to sugar-derived carbodiimides has been examined. Acetic acid efficiently catalysed the formation of ureas, whereas silica gel was found to be a more convenient catalyst in the case of the thioxo analogues. The procedures have been exploited in the development of an amine- and isocyanate-free synthesis of urea- and thiourea-tethered pseudooligosaccharides via the corresponding glycosylcarbodiimido sugars. The fully unprotected compounds adopted, preferentially, the (Z,Z) configuration at the pseudoamide bonds in water solution.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminoglycosides
  • Anti-Bacterial Agents / chemistry
  • Carbodiimides / chemistry*
  • Carbohydrate Conformation
  • Glycosides / chemical synthesis
  • Glycosides / chemistry*
  • Molecular Mimicry
  • Nuclear Magnetic Resonance, Biomolecular
  • Solutions
  • Stereoisomerism
  • Thiourea / analogs & derivatives*
  • Thiourea / chemical synthesis
  • Thiourea / chemistry
  • Water

Substances

  • Aminoglycosides
  • Anti-Bacterial Agents
  • Carbodiimides
  • Glycosides
  • Solutions
  • Water
  • Thiourea