Replacement of glycine 232 by aspartic acid in the KdpA subunit broadens the ion specificity of the K(+)-translocating KdpFABC complex

Biophys J. 2000 Aug;79(2):802-13. doi: 10.1016/S0006-3495(00)76337-5.

Abstract

Replacement of glycine residue 232 with aspartate in the KdpA subunit of the K(+)-translocating KdpFABC complex of Escherichia coli leads to a transport complex that has reduced affinity for K(+) and has lost the ability to discriminate Rb(+) ions (, J. Biol. Chem. 270:6678-6685). This glycine residue is the first in a highly conserved GGG motif that was aligned with the GYG sequence of the selectivity filter (P- or H5-loop) of K(+) channels (, Nature. 371:119-122). Investigations with the purified and reconstituted KdpFABC complex using the potential sensitive fluorescent dye DiSC(3)(5) and the "caged-ATP/planar bilayer method" confirm the altered ion specificity observed in uptake measurements with whole cells. In the absence of cations a transient current was observed in the planar bilayer measurements, a phenomenon that was previously observed with the wild-type enzyme and with another kdpA mutant (A:Q116R) and most likely represents the movement of a protein-fixed charge during a conformational transition. After addition of K(+) or Rb(+), a stationary current could be observed, representing the continuous pumping activity of the KdpFABC complex. In addition, DiSC(3)(5) and planar bilayer measurements indicate that the A:G232D Kdp-ATPase also transports Na(+), Li(+), and H(+) with a reduced rate. Similarities to mutations in the GYG motif of K(+) channels are discussed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphatases / chemistry*
  • Adenosine Triphosphatases / metabolism*
  • Amino Acid Sequence
  • Amino Acid Substitution
  • Aspartic Acid*
  • Carrier Proteins / chemistry*
  • Carrier Proteins / metabolism*
  • Cation Transport Proteins*
  • Cell Membrane / physiology
  • Cell Membrane / ultrastructure
  • Escherichia coli / physiology
  • Escherichia coli Proteins*
  • Glycine*
  • Kinetics
  • Lipid Bilayers
  • Liposomes
  • Macromolecular Substances
  • Membrane Potentials
  • Models, Molecular
  • Molecular Sequence Data
  • Potassium / metabolism*
  • Protein Conformation
  • Proteolipids / chemistry
  • Proteolipids / metabolism
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism

Substances

  • Carrier Proteins
  • Cation Transport Proteins
  • Escherichia coli Proteins
  • Lipid Bilayers
  • Liposomes
  • Macromolecular Substances
  • Proteolipids
  • Recombinant Proteins
  • proteoliposomes
  • Aspartic Acid
  • Adenosine Triphosphatases
  • potassium translocating Kdp-ATPase, E coli
  • Potassium
  • Glycine