Androgen and estrogen receptors in splenic T lymphocytes: effects of flutamide and trauma-hemorrhage

Shock. 2000 Oct;14(4):465-70. doi: 10.1097/00024382-200014040-00008.

Abstract

The endogenous sex steroids, testosterone and beta-estradiol, play a major role in inflammatory processes. They regulate several cytokine genes by interaction with their intracellular receptors that are, essentially, transcription factors. Because T-lymphocyte functions are altered following trauma-hemorrhage in male mice, we investigated whether (i) receptors for androgen (AR) and estrogen (ER) are present in splenic T lymphocytes, (ii) receptor expressions are altered following trauma-hemorrhage, and (iii) pretreatment of male mice with the AR antagonist, flutamide, alters receptor expressions and IL-6 release. Analysis of nuclear extracts indicated the presence of AR and ER in splenic T lymphocytes. No difference in receptor expressions between males and females or following trauma-hemorrhage was observed. Pretreatment of males with flutamide, however, led to increased ER expression in T lymphocytes of sham and trauma-hemorrhaged animals. This suggested that flutamide is capable of inducing the expression of another receptor belonging to a different gonadal steroid. Because response elements for AR and ER are present in the promoter region of the IL-6 gene, release of IL-6 and expression of signal transducer and activator of transcription 3 (STAT3) were analyzed as functional parameters in splenic T lymphocytes. Trauma-hemorrhage decreased IL-6 release by T lymphocytes and the release was restored to sham levels with flutamide pre-treatment. Similarly, STAT3 expression was decreased in T lymphocytes following trauma-hemorrhage and the expression was restored by flutamide pre-treatment. These data collectively demonstrate the importance of gonadal steroids in the regulation of splenic T-lymphocyte functions.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Androgen Antagonists / pharmacology*
  • Animals
  • DNA-Binding Proteins / metabolism
  • Female
  • Flutamide / pharmacology*
  • Hemorrhage / metabolism*
  • Interleukin-6 / metabolism
  • Male
  • Mice
  • Mice, Inbred C3H
  • Receptors, Androgen / drug effects*
  • Receptors, Androgen / metabolism*
  • Receptors, Estrogen / drug effects*
  • Receptors, Estrogen / metabolism*
  • STAT3 Transcription Factor
  • Sex Characteristics
  • Spleen / cytology
  • Spleen / drug effects
  • Spleen / metabolism
  • T-Lymphocytes / drug effects*
  • T-Lymphocytes / metabolism*
  • Testosterone / blood
  • Trans-Activators / metabolism
  • Wounds and Injuries / metabolism*

Substances

  • Androgen Antagonists
  • DNA-Binding Proteins
  • Interleukin-6
  • Receptors, Androgen
  • Receptors, Estrogen
  • STAT3 Transcription Factor
  • Stat3 protein, mouse
  • Trans-Activators
  • Testosterone
  • Flutamide