Neurotoxic regimen of methamphetamine produces evidence of behavioral sensitization in the rat

Synapse. 2001 Jan;39(1):1-7. doi: 10.1002/1098-2396(20010101)39:1<1::AID-SYN1>3.0.CO;2-7.

Abstract

A neurotoxic regimen of methamphetamine (MA) produces long-term depletions in neostriatal dopamine and serotonin concentrations. In addition to evidence of dopaminergic and serotonergic neurotoxicity, there is evidence of MA-induced behavioral changes. In this regard, stereotypic behavior elicited by MA is greater in rats treated previously with a neurotoxic regimen of MA than in control animals. The present study was designed to determine whether the enhanced stereotypy observed in MA-treated rats is due to the MA-induced loss of dopamine (neurotoxicity) or to the repeated exposure to MA (sensitization). Rats were treated with MA (10 mg/kg every 2 h for four injections) or vehicle at either a normal (24 degrees C) room temperature or a cold (4 degrees C) room temperature, which has been shown to attenuate the MA-induced loss of dopamine. Stereotypy was assessed 7 days after treatment. Rats that had received a neurotoxic regimen of MA at 24 degrees C exhibited 49% and 45% reductions in neostriatal dopamine and serotonin concentrations, respectively, whereas rats treated with MA at 4 degrees C had no significant neurochemical depletions. Stereotypy elicited by MA (5.0 mg/kg) was significantly greater in rats treated with a neurotoxic regimen of MA regardless of the initial treatment temperature. In addition, an injection of apomorphine (0.5 mg/kg) elicited an enhanced stereotypic response in MA-treated rats. These data suggest that the augmented stereotypic behavior observed in rats treated with a neurotoxic regimen of MA is not due to the loss of dopamine, but rather the manifestation of behavioral sensitization, possibly due to an increase in dopamine receptor sensitivity.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Apomorphine / pharmacology
  • Brain / cytology
  • Brain / drug effects*
  • Brain / metabolism
  • Cold Temperature / adverse effects
  • Dopamine / metabolism
  • Male
  • Methamphetamine / toxicity*
  • Neostriatum / cytology
  • Neostriatum / drug effects
  • Neostriatum / metabolism
  • Neurons / cytology
  • Neurons / drug effects*
  • Neurons / metabolism
  • Neurotoxins / toxicity*
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Dopamine / drug effects
  • Receptors, Dopamine / metabolism
  • Serotonin / metabolism
  • Stereotyped Behavior / drug effects*
  • Stereotyped Behavior / physiology

Substances

  • Neurotoxins
  • Receptors, Dopamine
  • Serotonin
  • Methamphetamine
  • Apomorphine
  • Dopamine