p38 mitogen-activated protein kinase regulates low potassium-induced c-Jun phosphorylation and apoptosis in cultured cerebellar granule neurons

J Biol Chem. 2001 Feb 16;276(7):5129-33. doi: 10.1074/jbc.M007258200. Epub 2000 Nov 16.

Abstract

Cultured rat cerebellar granule neurons are widely used as a model system for studying neuronal apoptosis. After maturation by culturing in medium containing 26 mm potassium (high K(+)), changing to medium containing 5 mm potassium (low K(+); LK) rapidly induces neuronal apoptosis. Then over 50% of granule cells die within 24 h. However, the molecular mechanisms by which the LK-induced apoptosis occurs in cultured cerebellar granule cells remain unclear. In the present study, we found that p38 MAP kinase (p38) was an important factor for LK-induced apoptosis. Three hours after changing to LK medium, p38 was markedly activated. In addition, SB203580, a specific inhibitor of p38, strongly inhibited the phosphorylation and expression of c-Jun in LK-induced apoptosis of cultured cerebellar granule cells. In vitro kinase assay using glutathione S-transferase-c-Jun as a substrate showed that p38 directly phosphorylated c-Jun. Furthermore, in the presence of SB203580, about 80% of neurons survived. These results indicate that p38 regulates LK-induced apoptosis of cerebellar granule neurons.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis* / drug effects
  • Cells, Cultured
  • Cerebellum / metabolism
  • Enzyme Activation
  • Enzyme Inhibitors / pharmacology
  • Imidazoles / pharmacology
  • Kinetics
  • Mitogen-Activated Protein Kinases / physiology*
  • Neurons / cytology*
  • Neurons / drug effects
  • Neurons / metabolism
  • Phosphorylation
  • Potassium / pharmacology*
  • Proto-Oncogene Proteins c-jun / metabolism*
  • Pyridines / pharmacology
  • Rats
  • Rats, Wistar
  • p38 Mitogen-Activated Protein Kinases

Substances

  • Enzyme Inhibitors
  • Imidazoles
  • Proto-Oncogene Proteins c-jun
  • Pyridines
  • Mitogen-Activated Protein Kinases
  • p38 Mitogen-Activated Protein Kinases
  • SB 203580
  • Potassium