Mutations conferring ganciclovir resistance in a cohort of patients with acquired immunodeficiency syndrome and cytomegalovirus retinitis

J Infect Dis. 2001 Jan 15;183(2):333-337. doi: 10.1086/317931. Epub 2000 Dec 15.

Abstract

Cytomegalovirus (CMV) retinitis is among the most common opportunistic infections in patients with acquired immunodeficiency syndrome. In a prospective study of 210 patients with CMV retinitis, 26 were identified as having either a phenotypic or a genotypic ganciclovir-resistant isolate from either blood or urine cultures. For blood culture isolates with an IC(50) >6.0 microm for ganciclovir, the sensitivity and specificity for detecting a UL97 mutation were 95% and 98%, respectively, whereas for an IC(50) >8.0 microM they were 79% and 99%, respectively. Although there were trade-offs between the 2 thresholds for blood culture isolates, for urine culture isolates an IC(50) >8.0 microM appeared to be better at identifying genotypic resistance. UL97 mutations identified in both the blood and urine cultures of individual patients were identical in 87.5% of cases. High-level ganciclovir resistance (IC(50), >30 microM) typically, but not invariably, was associated with a mutation in both the UL97 and UL54 genes.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • AIDS-Related Opportunistic Infections / virology*
  • Adult
  • Aged
  • Antiviral Agents / pharmacology*
  • Blood / virology
  • Cohort Studies
  • Cytomegalovirus / drug effects*
  • Cytomegalovirus / genetics
  • Cytomegalovirus / isolation & purification
  • Cytomegalovirus Retinitis / virology*
  • DNA-Directed DNA Polymerase / genetics
  • Drug Resistance, Microbial / genetics
  • Female
  • Ganciclovir / pharmacology*
  • Genotype
  • Humans
  • Male
  • Middle Aged
  • Mutation*
  • Phenotype
  • Phosphotransferases (Alcohol Group Acceptor) / genetics
  • Prospective Studies
  • Urine / virology
  • Viral Proteins*

Substances

  • Antiviral Agents
  • UL54 protein, Human herpesvirus 5
  • Viral Proteins
  • Phosphotransferases (Alcohol Group Acceptor)
  • ganciclovir kinase
  • DNA-Directed DNA Polymerase
  • Ganciclovir