Therapeutic effects of an oral adsorbent on acute dextran sulphate sodium-induced colitis and its recovery phase in rats, especially effects of elimination of bile acids in gut lumen

Dig Liver Dis. 2000 Nov;32(8):691-8. doi: 10.1016/s1590-8658(00)80332-1.

Abstract

Background: The pathogenesis of inflammatory bowel disease is still unknown. However, it is possible that faecal bile acids influence the clinical course.

Aims: To evaluate the eliminating effects of faecal bile acids by the oral adsorbent on dextran sulphate sodium-induced rat colitis.

Methods: Rats were given 3% dextran sulphate sodium aqueous solution for 7 days, with or without concomitant administration of oral adsorbent, or the rats were given dextran sulphate sodium for 7 days, followed with or without oral adsorbent for 5 days. Macroscopic and microscopic examinations of the colons and measurement of faecal bile acids were performed. The cytotoxicity of bile salts on Caco-2 cells was also evaluated.

Results: Oral adsorbent tended to attenuate the dextran sulphate sodium-induced colitis. Oral adsorbent was fairly effective in reducing faecal hyodeoxycholic acid concentration. A positive correlation was found between the size of the ulcer area and the faecal hyodeoxycholic acid concentration. In a cell culture study, cytotoxicity of bile acid was parallel with increasing hydrophobicity of the bile acid. However, hyodeoxycholate exhibited severe cytotoxicity, despite its hydrophilic properties.

Conclusions: Oral adsorbent tended to attenuate the dextran sulphate sodium-induced colitis and tended to promote the recovery process. It is possible that bile acids in the gut lumen influence the progression of dextran sulphate sodium-induced colitis and its repair process.

MeSH terms

  • Acute Disease
  • Adsorption
  • Animals
  • Bile Acids and Salts / metabolism*
  • Bile Acids and Salts / pharmacology
  • Caco-2 Cells
  • Carbon / pharmacology*
  • Cell Survival / drug effects
  • Colitis / chemically induced
  • Colitis / drug therapy*
  • Colitis / pathology
  • Colitis / physiopathology*
  • Dextran Sulfate
  • Feces / chemistry
  • Humans
  • Inflammatory Bowel Diseases
  • Intestinal Mucosa / metabolism*
  • Male
  • Models, Animal
  • Oxides / pharmacology*
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Bile Acids and Salts
  • Oxides
  • Carbon
  • Dextran Sulfate
  • AST 120