The direct effect of IL-12 on tumor cells: IL-12 acts directly on tumor cells to activate NF-kappaB and enhance IFN-gamma-mediated STAT1 phosphorylation

Biochem Biophys Res Commun. 2001 Jan 19;280(2):503-12. doi: 10.1006/bbrc.2000.4150.

Abstract

IL-12 directly acts on T cells and NK cells to induce IFN-gamma production. IFN-gamma plays an important role in anti-tumor effect of IL-12. In spite of various functions of IL-12 on immunocytes, the direct effect of IL-12 on tumor cells has not been fully clarified. The present study investigated the direct effect of IL-12 on eight murine tumor cell lines in vitro. IL-12 did not directly up-regulate expression of MHC class I on tumor cells, but enhanced IFN-gamma-induced up-regulation of MHC class I expression in MC-38, MCA102, MCA205 and MCA207 cells. IL-12 alone did not activate STAT1, but IL-12 enhanced IFN-gamma-mediated STAT1 phosphorylation in MC-38, MCA102, MCA205, MCA207 and Colon-26-NL-17 cells, which expressed IL-12 receptor beta1 mRNA. In the other side, Panc-02, B16-BL6 and 266-6 cells were not affected by IL-12, in which expression of IL-12 receptor beta1 mRNA was not detected. Anti-IL-12 mAb inhibited the direct effect of IL-12 on MC-38 cells. Moreover, nuclear localization of NF-kappaB was observed after stimulation of IL-12 or IL-12 p40 in MC-38 and Colon-26-NL-17 cells, but not in Panc-02 cells. These findings suggest that IL-12 directly acts on tumor cells through IL-12 receptor beta1 to activate NF-kappaB and enhance IFN-gamma-mediated STAT1 phosphorylation.

MeSH terms

  • Active Transport, Cell Nucleus / drug effects
  • Animals
  • Antibodies, Monoclonal / immunology
  • DNA / metabolism
  • DNA-Binding Proteins / metabolism*
  • Flow Cytometry
  • Histocompatibility Antigens Class I / metabolism
  • Interferon-gamma / metabolism
  • Interferon-gamma / pharmacology*
  • Interleukin-12 / agonists
  • Interleukin-12 / antagonists & inhibitors
  • Interleukin-12 / immunology
  • Interleukin-12 / pharmacology*
  • Mice
  • NF-kappa B / metabolism*
  • Phosphorylation / drug effects
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Receptors, Interleukin / metabolism
  • Receptors, Interleukin-12
  • STAT1 Transcription Factor
  • STAT4 Transcription Factor
  • Trans-Activators / metabolism*
  • Tumor Cells, Cultured
  • Up-Regulation / drug effects

Substances

  • Antibodies, Monoclonal
  • DNA-Binding Proteins
  • Histocompatibility Antigens Class I
  • Il12rb1 protein, mouse
  • NF-kappa B
  • RNA, Messenger
  • Receptors, Interleukin
  • Receptors, Interleukin-12
  • STAT1 Transcription Factor
  • STAT4 Transcription Factor
  • Stat1 protein, mouse
  • Stat4 protein, mouse
  • Trans-Activators
  • Interleukin-12
  • Interferon-gamma
  • DNA