Immediate and prolonged patterns of Agouti-related peptide-(83--132)-induced c-Fos activation in hypothalamic and extrahypothalamic sites

Endocrinology. 2001 Mar;142(3):1050-6. doi: 10.1210/endo.142.3.8018.

Abstract

Several lines of evidence substantiate the important role of the central nervous system melanocortin 3- and 4-receptor (MC3/4-R) system in the control of food intake and energy balance. Agouti-related peptide (AgRP), an endogenous antagonist of these receptors, produces a robust and unique pattern of increased food intake that lasts up to 7 days after a single injection. Little is known about brain regions that may mediate this powerful effect of AgRP on food intake. To this end we compared c-Fos-like immunoreactivity (c-FLI) in several brain sites of rats injected intracerebroventricularly with 1 nmol AgRP-(83--132) 2 and 24 h before death and compared c-FLI patterns to those induced by another potent orexigenic peptide, neuropeptide Y (NPY). Although both NPY and AgRP induced c-FLI in hypothalamic areas, AgRP also produced increased c-FLI in the accumbens shell and lateral septum. Although NPY elicited no changes in c-FLI 24 h after administration, AgRP induced c-FLI in the accumbens shell, nucleus of the solitary tract, central amygdala, and lateral hypothalamus. These results indicate that an NPY-like hypothalamic circuit mediates the short-term effects of AgRP, but that the unique sustained effect of AgRP on food intake involves a complex circuit of key extrahypothalamic reward and feeding regulatory nuclei.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Agouti-Related Protein
  • Animals
  • Brain / metabolism*
  • Hypothalamus / metabolism
  • Immunohistochemistry
  • Injections, Intraventricular
  • Male
  • Neuropeptide Y / pharmacology
  • Peptide Fragments / pharmacology*
  • Proto-Oncogene Proteins c-fos / physiology*
  • Rats
  • Rats, Long-Evans
  • Time Factors
  • Tissue Distribution / drug effects

Substances

  • Agouti-Related Protein
  • Neuropeptide Y
  • Peptide Fragments
  • Proto-Oncogene Proteins c-fos
  • agouti-related protein-(83-132)