Pharmacokinetics of enrofloxacin after intravenous and intramuscular administration in Angora goats

Can J Vet Res. 2001 Jan;65(1):64-7.

Abstract

Pharmacokinetics and bioavailability of enrofloxacin were determined after single intravenous (IV) and intramuscular (IM) administrations of 5 mg/kg body weight (BW) to 5 healthy adult Angora goats. Plasma enrofloxacin concentrations were measured by high performance liquid chromatography. Pharmacokinetics were best described by a 2-compartment open model. The elimination half-life and volume of distribution after IV and IM administrations were similar (t1/2beta, 4.0 to 4.7 h and Vd(ss),1.2 to 1.5 L/kg, respectively). Enrofloxacin was rapidly (t1/2a, 0.25 h) and almost completely absorbed (F, 90%) after IM administration. Mean plasma concentrations of enrofloxacin at 24 h after IV and IM administration (0.07 and 0.09 microg/mL, respectively) were higher than the minimal inhibitory concentration (MIC) values for most pathogens. In conclusion, once-daily IV and IM administration of enrofloxacin (5 mg/kg BW) in Angora goats may be useful in treatment of infectious diseases caused by sensitive pathogens.

MeSH terms

  • Animals
  • Anti-Infective Agents / administration & dosage
  • Anti-Infective Agents / blood
  • Anti-Infective Agents / pharmacokinetics*
  • Biological Availability
  • Chromatography, High Pressure Liquid
  • Communicable Diseases / drug therapy
  • Communicable Diseases / veterinary
  • Cross-Over Studies
  • Enrofloxacin
  • Fluoroquinolones*
  • Goat Diseases / drug therapy
  • Goats / metabolism*
  • Half-Life
  • Injections, Intramuscular / veterinary
  • Injections, Intravenous / veterinary
  • Microbial Sensitivity Tests
  • Quinolones / administration & dosage
  • Quinolones / blood
  • Quinolones / pharmacokinetics*

Substances

  • Anti-Infective Agents
  • Fluoroquinolones
  • Quinolones
  • Enrofloxacin