Abstract
P22PRG1/IEX-1 is a putative NF-kappaB target gene implicated in the regulation of cellular viability. Here, we show that in HeLa cells TNFalpha induces expression of p22PRG1/IEX-1 in an NF-kappaB dependent fashion. Blockade of NF-kappaB activation by various NF-kappaB inhibitors abolished TNFalpha-induced p22PRG1/IEX-1 expression and increased the sensitivity to apoptosis induced by TNFalpha, an activating Fas-antibody or the anti-cancer drug etoposide. Surprisingly, ectopic expression of p22PRG1/IEX-1 in HeLa cells transfected with an inducible p22PRG1/IEX-1-expression vector augments the susceptibility to apoptosis initiated by death-receptor ligands or by etoposide. In addition, p22PRG1/IEX-1 expressing HeLa cells exhibit an accelerated progression through the cell cycle. Transfection of an antisense hammerhead ribozyme targeted to p22PRG1/IEX-1 reduced the speed in cell cycle progression and decreased the apoptotic response to death ligands. Our data demonstrate that p22PRG1/IEX-1 is specifically induced during NF-kappaB activation, but this seems not to be related to the anti-apoptotic actions of NF-kappaB. Instead, NF-kappaB dependent recruitment of p22PRG1/IEX-1 might be related to a modulation in the cell cycle, and hereby, p22PRG1/IEX-1 may accelerate cell growth on the one hand, but may trigger apoptosis on the other. Oncogene (2001) 20, 69 - 76.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Anti-Inflammatory Agents, Non-Steroidal / pharmacology
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Antineoplastic Agents / pharmacology
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Apoptosis / drug effects
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Apoptosis / genetics*
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Apoptosis Regulatory Proteins
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Cell Cycle / drug effects
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Cell Cycle / genetics
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Cell Death / genetics
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Genetic Vectors / metabolism
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Gliotoxin / pharmacology
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HeLa Cells / cytology*
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HeLa Cells / drug effects
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HeLa Cells / metabolism*
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Humans
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Hydrolysis
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Immediate-Early Proteins / biosynthesis*
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Immediate-Early Proteins / genetics*
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Immediate-Early Proteins / metabolism
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Immediate-Early Proteins / physiology
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Immunosuppressive Agents / pharmacology
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Leucine / analogs & derivatives*
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Leucine / pharmacology
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Leupeptins / pharmacology
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Membrane Glycoproteins / biosynthesis*
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Membrane Glycoproteins / genetics*
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Membrane Glycoproteins / metabolism
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Membrane Glycoproteins / physiology
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Membrane Proteins
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NF-kappa B / antagonists & inhibitors
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NF-kappa B / metabolism
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NF-kappa B / physiology*
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Neoplasm Proteins*
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RNA, Catalytic / metabolism
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Sulfasalazine / pharmacology
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Tetracycline / pharmacology
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Transfection
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Tumor Necrosis Factor-alpha / pharmacology
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Tumor Necrosis Factor-alpha / physiology
Substances
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Anti-Inflammatory Agents, Non-Steroidal
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Antineoplastic Agents
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Apoptosis Regulatory Proteins
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IER3 protein, human
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Immediate-Early Proteins
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Immunosuppressive Agents
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Leupeptins
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Membrane Glycoproteins
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Membrane Proteins
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NF-kappa B
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Neoplasm Proteins
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RNA, Catalytic
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Tumor Necrosis Factor-alpha
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acetyl-leucinal-leucinal-normethional
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Sulfasalazine
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Gliotoxin
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Tetracycline
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Leucine
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benzyloxycarbonylleucyl-leucyl-leucine aldehyde