Generation of human high-affinity antibodies specific for the fibroblast activation protein by guided selection

Eur J Biochem. 2001 Mar;268(6):1730-8.

Abstract

Four completely human antibody derivatives [single-chain-antibody fragments (scFvs)] with specificity for the general tumor stroma marker fibroblast activation protein (FAP) were isolated by guided selection. Highly diverse IgG, IgM and IgD isotypes comprising heavy-chain variable domain libraries were generated using cDNAs derived from diverse lymphoid organs of a multitude of donors. Three of the human scFvs were converted into bivalent minibodies and expressed in eukaryotic cells for further functional characterization. Binding-competition studies and analysis by fluorescence-activated cell sorting showed high-affinity binding (10--20 nM) for two clones and recognition of the same epitope as the murine guiding antibody. The minibodies were successfully used for immunohistology of a variety of human carcinoma biopsies, revealing specific staining of stromal fibroblasts. Therefore, they should be suitable for in vivo diagnostic and tumor-targeting studies and, because of their completely human origin, be superior to murine or humanized antibody derivatives.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Antibodies, Monoclonal / chemistry
  • Antibodies, Monoclonal / immunology*
  • Antigens, Neoplasm*
  • Base Sequence
  • Binding, Competitive
  • Biomarkers, Tumor*
  • DNA Primers
  • DNA, Complementary
  • Endopeptidases
  • Gelatinases
  • Growth Substances / chemistry
  • Growth Substances / immunology*
  • Humans
  • Immunohistochemistry
  • Membrane Proteins
  • Molecular Sequence Data
  • Neoplasms / immunology
  • Sequence Homology, Amino Acid
  • Serine Endopeptidases / chemistry
  • Serine Endopeptidases / immunology*

Substances

  • Antibodies, Monoclonal
  • Antigens, Neoplasm
  • Biomarkers, Tumor
  • DNA Primers
  • DNA, Complementary
  • Growth Substances
  • Membrane Proteins
  • Endopeptidases
  • Serine Endopeptidases
  • fibroblast activation protein alpha
  • Gelatinases